ZempiloAmalungiselelo

Drug "Valvira": Ukubuyekezwa oogqirha

Njani ichiza "Valvira"? Reviews ngale medicament inokufumaneka materials nqaku. Kwakhona, oko kuluhlu ezo ezibonisa ukuba ukusetyenziswa kweziyobisi, neziphumo zalo, Izimo kunye nangaphezulu.

Ubume, iziyobisi ezingxobeni nemilo yayo

Ziziphi fomu iveliswa ichiza "Valvira"? Ukuphonononga uxele ukuba olu nyango zingathengwa ngokohlobo a macwecwe emhlophe okweqanda biconvex, umboniso-camera. Le esisebenza yale arhente izenzo valacyclovir hydrochloride ukuphilisa. amacandelo Njengoko eyongezelweleyo ukusetyenziswa kweziyobisi ingqalelo microcrystalline neselulosi kunye povidone.

Ngokubhekiselele ifilimu ukutyabeka, ngoko iquka giproloza, Opadry emhlophe, titanium dioxide, hypromellose kunye Macrogol.

Medicament "Valvira", ncomo kuzo zidweliswe ngezantsi, oku kuthengiswa imiqulu blister ye-aluminiyam eneli kunye PVC, ezo zingafakwa kwiibhokisi kwikhadibhodi.

features kwemithi

Yintoni iimpawu ichiza "Valvira"? Izimvo oogqirha bathi ukuba i-arhente antiviral. Kanye valaciclovir emzimbeni womntu iguqulelwe ngoko nangoko L-valine kunye acyclovir. Oku kwenzeka phantsi kwempembelelo valatsiklovirgidrolazy.

iziyobisi kujongwa liveza umsebenzi ethile inhibitory nxamnye herpes simplex virus, varicella zoster, cytomegalovirus, njalo-njalo. D.

Acyclovir uyakwazi ukwehlisa le Yindibanisela DNA wentsholongwane egazini, kwakunye acyclovir triphosphate zaguqulelwa kwifom esebenzayo. Le nto ke ifakwe kwi-DNA viral, nto leyo ekugqibeleni kukhokelela uqhekeko epheleleyo umxokelelwane yayo ekwathintela ukuphindaphindeka wentsholongwane egazini.

Pharmacokinetics

Emva kokufumana valacyclovir kweziyobisi ngokungenamkhethe ezabalazela ngokukhawuleza ukusuka phecana zesisu. A idosi enye amacwecwe (0.25-2 g) ufikelela xiyimiso ubuninzi egazini kwisithuba seeyure 1-2. Ngaloo ndlela bioavailability beziyobisi yi 54%, kungakhathaliseki ukuba ukutya.

Unxibelelwano acyclovir plasma iphantsi yaye malunga ne-15%. Le into abelwa ngokukhawuleza kakhulu zonke izicwili. Izakufunyanwa kwi isibindi, intso, izihlunu kunye nemiphunga. Acyclovir kwakhona lingena singene ulwelo lwe-cerebrospinal, secretion langasese kunye vesicles herpetic.

Xa abantu nokusebenza okuqhelekileyo sezintso kupheliswe isiqingatha ubomi ichiza 3 HR. Valaciclovir kukhuthaza livela nomchamo.

Ubungqina obubonakalayo buxela

Enoba ayazazi iinjongo apho emiselwe ichiza "Valvira" (tablets)? Izimvo yeengcali abanamava aziswe okukhomba zilandelayo:

  • herpes zoster;
  • herpes labial;
  • izifo elikhala ye kwiinwebu nesikhumba (kuthintelo nonyango), zinto ezo zibangelwa yintsholongwane herpes simplex (kubandakanywa nezolo esanda kwafunyaniswa ukuba herpes zangasese);
  • cytomegalovirus HIV (prophylaxis), elavela ngexesha abohlukeneyo.

Kwakhona amayeza kubhekwe emiselweyo ukunciphisa usuleleko yeqabane herpes obuni obusempilweni ngexesha lokwabelana ngesondo. Nangona kunjalo, oku kufuneka kuthathwe ngoko unyango suppressive xa zidityaniswe kunye namanye amayeza (iikhondom kunye m. P.).

Izimo

Kwezinye iimeko, izigulane musa ukumisela amayeza "Valvira"? Imiyalelo kwakhona oogqirha bathi Izimo zilandelayo:

  • bone ngumongo abohlukeneyo;
  • uhlobo ngokwezonyango kakhulu zosulelo lwe-HIV;
  • yobudala yabantwana;
  • abohlukeneyo sezintso;
  • Hypersensitivity ku acyclovir, valacyclovir, kunye nezinye izinto iziyobisi.

Ngononophelo amayeza kakhulu emiselweyo kubantu abane hepatic (ingakumbi iidosi eziphezulu), ukusilela kwezintso, xa ukhulelwe kwaye ngexesha lokuncancisa.

Drug "Valvira": imiyalelo yokusebenzisa

Reviews ngale medicament kuya kuxoxwa ngezantsi.

Kufuneke njani iipilisi antiviral? Amayeza emiselweyo abadala ngaphakathi. Le yedosi ixhomekeke kuhlobo kunye nobungozi besi sifo.

  • Tile - 1000 mg kathathu ngemini iveki.
  • Herpes simplex - 500 mg kabini yonke imihla. Xa izinga zingabuyi unokuthatha iintsuku 3-5, yaye episode yokuqala - ukuya kwiintsuku ezili-10.
  • herpes Labial - 2 g amaxesha 2 ngosuku. Ithamo yesibini kufuneka kuthathwe kwiiyure ezili-12 kamva.
  • Uthintelo losuleleko nezolo, apho zibangelwa yi-herpes simplex virus kubantu abanamajoni abaqhelekileyo omzimba - 500 mg kanye ngemini, kunye sisifo rhoqo - 250 mg kabini yonke imihla kubantu abadala kunye intswelo omzimba - 500 mg kabini ngemini. Ubude unyango na iinyanga 5-12.
  • Uthintelo losuleleko cytomegalovirus kwi olufikisayo abangaphezu kweminyaka elishumi abadala - grams ezimbini kane ngemini. Ubude unyango iinyanga ezintathu.

Njengoko kuthintelo losulelo lwe neqabane esempilweni ukuba ichiza "Valvira" (1500) ukuba herpes? Iingcali Guest bathi abantu immunocompetent kunye likakade rhoqo amayeza ibhalwa isixa mg 500 kanye usuku lube ngunyaka. Xa izenzo non-rhoqo ngesondo iyeza kufuneka ziqalwe ngeentsuku ezintathu.

Ithamo kufuneka incitshiswe kwizigulane kunye kumsebenzi kidney kakuhle.

Amatyala libanda, iipilisi

Ziziphi iimpawu kwenzeka xa ukutya iziyobisi engalunganga "Valvira"? Izimvo kumagqirha zibonisa mpawu zilandelayo libanda: isicaphucaphu, ukudideka, ukugabha, ukusilela kwezintso, intloko ebuhlungu, ukunyuka serum creatinine yoxinaniso, nemibono, ukuxhuzula, ukuphazamiseka, ukuba khokhoma.

Amaxhoba kufuneka abe phantsi kweliso unyango rhoqo ukuze ukubona iziphumo ezinetyhefu ezi mpawu.

Ihaemodialysis ikuvumela ukuba ukususa ngokupheleleyo acyclovir egazini.

imiphumela emibi

reactions Yintoni icala kungenzeka izigulane abafumana "Valvira" ukulungiselela (500 mg). Izimvo izigulane ezininzi ngokufuthi sithetha iziphumo ezifana kunganqwenelekiyo ukuba zenzeke, ezifana isicaphucaphu kunye intloko ebuhlungu. Kwakhona ingqalelo neziyobisi kwaye baxabane icala kakhulu kakhulu ezifana purpura thrombotic thrombocytopenic, ukusilela etsolo kwezintso, hemolytic-uremic syndrome nokuphazamiseka luvo.

Ukongeza koku kungasentla, iingcali zithi, kunye neziphumo ezibi zilandelayo:

  • kabi esiswini;
  • leukopenia, thrombocytopenia;
  • anaphylaxis;
  • kukuphazamiseka, isiyezi, ukuphazamiseka, ukudakumba, ukudideka, iimpawu ngengqondo, nemibono, Encephalopathy, kwengqondo, dysarthria;
  • dyspnea;
  • irhashalala, photosensitivity, pruritus;
  • angioedema, urticaria;
  • nezitenxo kwezi kidney;
  • ukungaboni;
  • neutropenia, vasculitis leykoplastichesky, igazi aplastic, purpura thrombocytopenic, thrombotic;
  • erythema multiforme;
  • hypercreatininemia, kunciphisa umthamo;
  • izifo ezihlasela zosulele ngokuphefumla phecana, seTrojan, tachycardia, arthralgia, ukudinwa, nasopharyngitis, emzimbeni, ukudumba kobuso, ifiva, ukwanda koxinzelelo lwegazi, rhinorrhea.

iingcebiso ezithile lolwamkelo esikolweni "Valvira" drug (indlela ukuthatha: phambi kokutya okanye emva kokutya)?

Izimvo oogqirha bathi bioavailability beziyobisi izimele zokungenisa ukutya. Ngoko ke, oko kuthathwe omabini ngexesha sidlo nasemva. Eyona nto ibalulekileyo - ukujonga izithuba ngokulinganayo phakathi idosi yemihla ngemihla.

Kufuneka kuqatshelwe ukuba hlengiso Izikali abadala kuphela kungajongwangwa ntsingiselo, ngaphandle kwakwiimeko apho kukho nezitenxo ebalulekileyo kwizintso.

amava lwezonyango kunye beziyobisi abantwana abaselula engekhoyo. Ngoko ke, ukuba abele iintsana enjalo ichiza ongaphantsi kweminyaka 12-14 ayikhuthazwa.

Reviews imithi

Herpes - yintsholongwane zikukhathazayo abantu abaninzi ehlabathini lonke. Ngoko ke, "Valvira" ichiza kwemfuno enkulu kwimarike yezemithi. Ngokutsho iimpendulo lezigulane, eli yeza ikhuthaza ukupheliswa ngokukhawuleza yezilonda herpes, kwakunye nokuphuculwa isigulane kakuhle-ntle.

"Valvira" lisetyenziswa nje ukunyanga intsholongwane wathi, kodwa njengenyathelo lothintelo. Abantu abaninzi bathi xa ukuthatha eli amayeza nezihlandlo isahlakalo herpes leyo kakhulu lifinyele.

Asikwazi bathi ukuba yonke imigaqo yokuthatha amayeza, oko phantse zange zibangele ukuba ngaba iziphumo ebezingalindelekanga. Nakuba kunjalo, kufanele kuqatshelwe ukuba kunye nengxelo ngokuqhubekayo ethembisa kakhulu evela kweli chiza nazo negative. ukuba abaninzi kubo ezinxulumene yexabiso eliphezulu ichiza. Okwangoku, tablets ezilishumi (500 mg) "Valvira" zingathengwa ngenxa 600-680 engange.

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