Ichiza "Ksarelto" imiyalelo zokusetyenziswa njengendlela elichaza, yinto anticoagulant yesenzo ngqo. Xa isiseko sesi ichiza a inhibition ngqo factor nagyo. Ngaphaya koko, eli chiza a selectivity eliphezulu. Ke ukuba pharmacokinetics yayo, oko ako ngokukhawuleza kakhulu, afikelele xiyimiso ophezulu egazini emva kweeyure nje ezimbini ukuya kwezine emva kulawulo ngomlomo. Ukuba sithethe malunga iimpawu zinomgutyulo ophezulu ichiza, kunye umchamo kunye ndle eboniswe malunga 92-95% amayeza "Ksarelto". Imiyalelo yokusebenzisa (ixabiso, ngasendleleni, oku kuthetha ukuba malunga 1500 engange) kuqatshelwe apha ukuba inxalenye eseleyo ushiya umzimba ngohlobo kutshintsha yi zinomgutyulo kwezintso.
Efumanekayo le anticoagulant ngohlobo amacwecwe ngeenxa epinki emnyama okanye umbala obomvu-omdaka, equlethe kumafa zalo ezilishumi, elinesihlanu okanye amashumi amabini neemiligram rivaroxaban micronized. Nezincedisi-mzimba zizinto ezifana croscarmellose isodiyam, isodiyam lauryl sulfate, hypromellose 5cP, microcrystalline kwincindi, nemagnesium stearate kunye monohydrate lactose. Ekwakhiweni shell iquka titanium dioxide, Macrogol 3350 kunye ne-nitric ferric ebomvu. Ukongeza, umthamo omncinane iqulethe hypromellose 5cP.
Misa pill "Ksarelto" imiyalelo zokusetyenziswa ekucetyiswa ngokubanzi izigulane abaye ngaphambili ukufumene iinkqubo zotyando eziphelweni asezantsi. Kuba didi lwabantu isenzo anticoagulant njengenyathelo oluphumelelayo lokunqanda ukuba kuphuhliso lwexesha elizayo thromboembolism lwemithambo. Ukongeza, ichiza "Ksarelto" ngokugqibeleleyo ezifanelekileyo ukunqanda ukuphinda DVT kunye PE. Kwakhona, esi sixhobo kufuneka isetyenziselwe nokuthintela icala kubantu abane fibrillation atrial, uhlobo non-valvular. Ukuthintela uphuhliso thromboembolism lwenkqubo kunye nonyango lwe thrombosis ndlela olunzulu occlusion yayiyazi loo pulmonary kwakhona icebisa ukuba uthatha iipilisi "Ksarelto" umyalelo manual.
Sebenzisa le anticoagulant nto contraindicated ngqongqo kubantu abane emathunjini, intracranial okanye naziphi na ezinye iintlobo ukopha, i kakhulu lwe ukusilela kwezintso nobandlululo ku galactose. Kwimeko hypersensitivity isigulane ukuba rivaroxaban okanye uxabane kwezinye excipients kuluhlu ekwakhiweni, kwaye kufuneka bathathe amachiza "Ksarelto". Imiyalelo yokusebenzisa uyakuthintela kulimisela ngamandla kwaye ngexesha lokukhulelwa. Izimo nabo lactose akaxoleli, unyango kunye nezinye anticoagulants, izifo zesibindi, ekhatshwa coagulopathy, kunye neemeko ezinxulumene emngciphekweni omkhulu nokopha. Ukongeza, awukwazi ukuthatha abafazi amayeza, mame, kunye nabantu ayifikanga kweminyaka elishumi elinesibhozo.