Zempilo, Amalungiselelo
Ngeempumlo spray "Dezrinit": reviews oogqirha, imiyalelo esetyenziswa kunye nokwakheka
"Dezrinit" - glucocorticosteroid eyenziweyo (GCS) isicelo mlonyeni. Iarhente esebenzayo yi mometasone antiallergic kunye antiinflammatory amanyathelo. Ekusebenziseni ichiza avumelekile ukuba ndingamkhubekisi iziphumo zenkqubo kombisa anti-ukudumba umsebenzi wayo mlonyeni. Qwalasela eli nqaku malunga "Dezrinit" impendulo ukulungiselela kumagqirha kunye nabathengi.
Ichiza kangako ukukhululwa yabalamli ukudumba, lipomodulin ekwandiseni imveliso, i inhibitor of phospholipase A, yaye oku kubangelwe wokwehla wakhululwa CD acid kunye prostaglandin amagama inhibition kunye endoperoxides elibujikele. Ichiza kukuthintela beqokelela neutrophils, ukunciphisa imveliso exudate yokukrala kunye lymphokine, inhibition zemfuduko macrophage, ukunciphisa iinkqubo granulation idibane, ukunciphisa ukuyilwa chemotaxis, okt nefuthe basabela kamva komzimba kwenzeka ukumisa uphuhliso basabela nangoko nawo.
Oku kuqinisekiswa kwi medicament "nohlolo Dezrinit 'loogqirha - abaziingcali intsimi yabo. Isakhiwo kuthetha iquka mometasone furoate kunye nezincedisi.
Pharmacokinetics
isicelo Intranasal kunciphisa bioavailability lwenkqubo mometasone furoate ukuya ngaphantsi kwe-1%. into esebenzayo nako ukungena egazini, hi mpimo lowutsongo wendele ngenkuthalo biotransformed emva yokupasa lokuqala esibindini. Kwi yokulungiselela "Dezrinit" Oogqirha review becala HIV.
Ngaba eboniswe:
- ukuphathwa kwabantwana nokuthimliswa komzimba ezikhula ngamaxesha ukusuka kwiminyaka-2 nangaphezulu abadala;
- sinusitis etsolo, exacerbation of sinusitis abantwana ezingapheliyo kweminyaka elishumi ubudala nangaphezulu, kunye nabantu abadala (kubandakanywa abadala) njenge unyango adjuvant kunye antibiotics;
- Unyango adenoids ebantwaneni okanye abadala polyposis ngeempumlo;
- uthintelo nokuthimliswa ngamaxesha komzimba kwiimeko aphakathi kwaye yababuhlungu abantwana ukusuka kwiminyaka elishumi ubudala nangaphezulu kwakunye nabantu abadala. YokuziPhatha Kucetyiswa ukuba kwiiveki ezine phambi kokuba kuqale dusting lonyaka.
release Form
spray ngeempumlo nogesi. Enye isitsha iqulethe amathamo 140. Ifom reference beziyobisi ngohlobo amathontsi ayisekho ngexesha lokulungiselela ncwadi. Ifanele "Dezrinit" abantwana. Izimvo oogqirha, siyandingqinela ukuba andixoki.
Indlela yokusebenzisa kunye nemiyalelo yokusebenzisa
Ichiza iphethwe intranasally. Spray equlethwe igutyana leyo lesitofu impumlo usebenzisa isixhobo okhethekileyo nomthamo.
Phambi kokuqala isicelo wesipreyi ukwenza kwiimpompo 10 uvavanyo kwi kwisixhobo nomthamo. Emva ekulinganisweni, umlinganiselo unikezelo amayeza icwangcisiwe, cinezela ngalinye uqengqa zokumiswa 100 mg leyo eziqulathwe 50 mcg of mometasone. Ngaphambi usebenzisa imveliso emva ngaphezu kokuba ikhefu imini-14, kunye nesandi sidlalwe kufuneka uphindaphindwe. Isicelo ngasinye kufuneka sikhatshwe yayibhekisela ishukumisa igutyana.
imiphumela emibi
About "Dezrinit» Amalungiselelo ncomo zonyango bacebisa ezi ziphumo zilandelayo ecaleni okunokwenzeka:
- glaucoma;
- reactions hypersensitivity kuquka dyspnea, kunye bronchospasm;
- anaphylaxis;
- ebuhlungu abantwana nabantu abadala;
- angioedema;
- nokopha;
- avuthayo lweHo- ngeempumlo;
- abantwana babe ukukhula efanele, lengqondo ukungahlaliseki, zokulala, ixhala, ukuziphatha silwe, ukudandatheka;
- umqala obuhlungu;
- perforation le zekhala ngeempumlo ;
- imvakalelo aphazamiseke le imazi ibonakalisa em- ngeempumlo;
- kuyabuya ukuluma isifo pharyngeal;
- izifo zangentla ezihlasela zosulele ngokuphefumla iphecana;
- uthimla;
- kungcamla ukuphazamiseka;
- ephula Isivamvo sokujoja;
- cataract;
- noxinzelelo intraocular;
- izilonda le isifo em- ngeempumlo.
Izimo
"Dezrinit" Drug (reviews of oogqirha ukuliqinisekisa) liyahlonyelwa contraindicated ku:
- hypersensitivity ku mometasone okanye naliphi na kumacandelo kuqulunqo;
- .. Ungenelelo ngotyando yakutshanje okanye ngeempumlo umothuko esilondeni impiliso, ukuba isinyathelo GCS ngendlela inhibitory kwi iinkqubo ephilisa;
- kubantwana (ukuba polyposis ngeempumlo 18; exacerbations nokoyika sinusitis esinganyangekiyo, oyingozi okanye ukuya kutsho kwiminyaka eli-12; abaneminyaka 2 nokuthimliswa kunye nee ezikhula ngamaxesha athile).
Ukusetyenziswa kweziyobisi ngethuba lokukhulelwa nokuncancisa
Ingakumbi akukho izifundo yokusetyenziswa ekhuselekileyo "Dezrinita" ngethuba lokukhulelwa lokwaphusa lwenziwa. Eli chiza kufuneka kwenziwa ngabo lokuncancisa kunye nabasetyhini abakhulelweyo kuphela xa izibonelelo impilo kamama wodlula nobungozi ukuba usana okanye olungekazalwa. Kubelekwa omama kusetyenziswa corticosteroids ngethuba lokukhulelwa, kufuneka bapase uviwo ekhethekileyo ukuchonga kunokwenzeka hypoadrenalism. Oku kuqinisekiswa kwi medicament "Dezrinit" uhlaziyo zizifo ezithile zonyango.
Ukusetyenziswa kweziyobisi for abantwana
Ukusetyenziswa "Dezrinita" into contraindicated ebantwaneni kunye ngeempumlo polyposis umgodi 18; i exacerbation of sinusitis ezinganyangekiyo okanye uhlobo nokoyika kwiminyaka ukuya ku-12; kunye nokuthimliswa ezikhula ngamaxesha bayaliwa kwiminyaka emi-2. Wayedla "Dezrinit" kwi adenoids ebantwaneni. Izimvo oogqirha kule nkalo ezincomekayo.
imiyalelo yokusebenzisa
Iimpawu ze yoma le isifo ngeempumlo emva unyango (iinyanga ezili-12) ngonyaka omnye zange ulandelwe. Uhlolisiso biopsies of isifo ngeempumlo abonisa ifuthe mometasone ukuba isimo kuqheleke histology. ukusetyenziswa kwexesha elide ichiza, kwakunye naluphi na unyango ixesha elide, kubandakanya uhlolo ngamaxesha ngeempumlo isifo igqirha otorhinolaryngology.
Xa nesifo umgudu (elele okanye esebenzayo); yintsholongwane, systemic viral (kubandakanywa herpes luchaphazela amehlo, okanye Herpes simplex) okanye ezinzwaneni; unyango elide ngu corticosteroids; ubukho usulelo olunganyangwanga lwasekhaya isifo ngeempumlo, kwakunye lokuncancisa kunye nokukhulelwa, ichiza kufuneka umisele ngononophelo.
Unyango lithetha "Dezrinit" yaleza ukuba uyeke kwaye uqale ukuqhuba unyango eyodwa kuphuhliso ezinzwaneni yasekuhlaleni pharynx okanye impumlo.
Kwinwebu pharynx nakumarhanana, leyo sithatha ixesha elide kakhulu kwexesha, kube njengento inkomba ukungaphumeleli ichiza. Unako kwakhona uqaphele ukuba akukho yatyhilwa kwezithandani kwenkqubo hypothalamic-yebhinqa-adrenal emva ukusetyenziswa elide ichiza. Oku kungqinwa ncomo elungiswa "Dezrinit".
ingqalelo ekhethekileyo ngokwayo ifuna izigulane zifumana unyango elide kunye corticosteroids, ngokugqithisela unyango kunye mometasone. Ukuba umisa GCS inkqubo intshukumo, ngoko ithuba sinokuthi oko kuya kubangela kukungabi umsebenzi adrenal, unyango leyo eza kufuna amanyathelo afanelekileyo.
Kwezinye izigulane, kwinguqu esa unyango mometasone emva corticosteroids Inokwenzeka uyeka ukusetyenziswa lwenkqubo glucocorticosteroids. Ezi ziquka ukudakumba, ukudinwa, iintlungu zezihlunu kunye / okanye amalungu. Izigulane kufuneka ezizodwa ukweyisela ukuba unyango with "Dezrinit" kufanelekile, nangona ukuhla ubungqongqo iimpawu izitshanguba isifo ngeempumlo. Zigqunyiweyo (kodwa sele sikhona kakade kumguli) unyango lwezifo glucocorticoid systemic komzimba ezifana nangokhwekhwe conjunctivitis, unako kuchongwa kunye lenguqu ukuya corticosteroids zasekuhlaleni.
Xa unyango polyp unilateral; polyp, zinxulunyaniswa abanesigulo esinganyangekiyo, kunye polyp, nesigubungelo ngokupheleleyo lweHo- ngeempumlo, ukhuseleko kunye nokusebenza kwe "Dezrinita" alikhange kufundwe. Ukopha kunye polyp unilateral ukuba i imilo mgaqweni, kuyimfuneko ukuphanda ngakumbi.
Izigulane zifumana unyango ngu corticosteroids, ufumane reactivity omzimba sinciphile kwaye ngoko kufuneka alumkise ukuba konyusa ingozi yosulelo ngokudibana yimasisi abagulayo, irhashalala kunye nezinye uhlobo ezosulelayo esi sifo, kwaye kufanele ubuze oyingcaphephe, ukuba kumfowunelwa isigulane kunjalo I zenzeka.
ukusetyenziswa elide corticosteroids ngeempumlo ngeedosi ezinkulu oluphenthwe kuphuhliso neziphumo ebezingalindelekanga. Nangona kunjalo, ezi ziphumo kuba kude ngaphantsi okuba ngaphezu xa corticosteroids systemic asetyenziswa, kwaye bayashiyana izigulane ngamnye. imiphumela systemic bazo ziquka syndrome Cushing, nto leyo luphawulwa ingcinezelo adrenal, glaucoma, cataract, abazizidalwa ngokukhula abantwana nabo bakwishumi elivisayo, kwaye maxa wambi eziliqela neziphumo zokuziphatha nangokwasengqondweni, kuquka ixhala, ukuphazamiseka ekulaleni, ukudakumba okanye ndlongo, lengqondo ukungahlaliseki.
Njengoko kuba intsebenziswano kweziyobisi phakathi iziyobisi ezahlukeneyo kunye mometasone, malunga olu phando lwenziwa.
Ngeempumlo spray «Teva Dezrinit": ncomo zabathengi kunye noogqirha
Izimvo zamalungiselelo becala ezintle. uncedo ezilungileyo nokuthimliswa komzimba. Ngesiqhelo ukunyamezeleka enqabile ukunika iziphumo ebezingalindelekanga. Abantwana abancinane kunceda adenoids, kunciphisa komtshiso oko. Eyona nto ibalulekileyo ukuba ukuhlonipha imiyalelo ukusetyenziswa.
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