Zempilo, Amalungiselelo
Ichiza "dopegit": Ukubuyekezwa oogqirha
Kuyanceda kuzinziswe ichiza "dopegit" xinzelelo. Izimvo kumagqirha besithi ayasebenza ngokukhawuleza nangendlela efanelekileyo. Kuyinto ayibizi. Kuthengiswa phantse yonke ekhemisti. Kuvumelekile ukuba athathwe yi abafazi abakhulelweyo. Iyeza iye Izimo, ngoko ke akukho mfuneko yokuba usele ngaphandle kagqirha.
Isakhiwo kunye Nokuhlanganiselwa
Drug "dopegit" (iimpendulo leengcali kuqinisekisa ukuba le unyango kuphela uxinzelelo yeminikelo ilungiselelwayo abasetyhini abakhulelweyo kunye lwegazi) ifumaneka emacwecweni. Ezi pilisi amhlophe, umbala nombala kancinane. Iqulethe malunga 282 mg esisebenza - methyldopa sesquihydrate. Le ubungakanani efanayo 250 mg methyldopa. Awongeziweyo amaqela amacwecwe zezi:
- amabele starch;
- stearic acid;
- talc;
- sodium carboxymethyl starch;
- ethyl neselulosi;
- wemagniziyam stearate.
Amacwecwe zahlanganiswa iibhotile zeglasi emnyama lamaqhosha mahlanu. Le imiyalelo apha ngenjongo yokuba uyisebenzise.
Isenzo amayeza ye ichiza
Jonga Wegetotropona antihypertensives central intshukumo "dopegit" iipilisi (iirivyu zonyango abasebenzi bathi eli yeza, amabhinqa amaninzi asele ngexesha lokukhulelwa). Xa emzimbeni, le medicament aguqulwa kwi metilnoradrenalina indalo alpha weklayenti isiphumo iqinile ngokwenza iindlela eziliqela. Ichiza kunciphisa ithoni novelwano. Oku kungenxa ipoti ye-ezinkulu inhibitory presynaptic .alpha.2-receptor.
Iyeza lisebenza njenge neurotransmitter lobuxoki nawethutyana, phezu kwalapho of dopamine dopaminergic iqala. Kunciphisa umsebenzi renin egazini kunye nomphumela ofanayo iyonke ukumelana peripheral. Kumisa Yindibanisela noradrenaline. Kunciphisa ukuyilwa epinephrine, dopamine, norepinephrine kunye serotonin ngenxa kwezithandani lwe umsebenzi enzyme dopa-decarboxylase.
Le into esebenzayo - methyldopa - aluchaphazeli intliziyo nomzimba yomsebenzi akuthethi ukunciphisa imveliso intliziyo. Musa ukusiphikisa imbonakalo tachycardia reflex. Ayichaphazeli isantya product glomerular. Akukho ukusebenza ngomhla igazi kwezintso kwaye akukho uxinzelelo iqhezu filterable.
Maxa wambi xa ukuthatha amayeza ukuze ukunciphisa izinga intliziyo. Amayeza kunciphisa ngokukhawuleza uxinzelelo lwegazi. Kwiimeko ezinqabe kakhulu, kunokubangela hypotension postural.
Emva amacwecwe kwedosi yokuqala enempembelelo enkulu emsebenzini emva kweeyure 4-6 kwaye sihlala iiyure ezili-12 ukuya kuma-24. Ichiza nga ukunciphisa uxinzelelo kwi ngosuku lwesibini okanye lwesithathu ukuthatha iipilisi.
ubungqina
Iimpawu zibonisa ukuba ukusetyenziswa "dopegit" iziyobisi (reviews athi ichiza akukho ngxaki unako ukuthenga kuyo nayiphi na ivenkile) yi lwegazi. Olu nyango lidla emiselweyo kwizigulane abakhulelweyo.
Izimo ukuba ukusetyenziswa kweziyobisi
Uphawula ukuba inika isiphumo ezilungileyo "dopegit" xi iziyobisi, ncomo zonyango. Ngaphandle koku, ichiza ungamiselwanga kohlobo kwinqanaba etsolo zophuhliso, zesibindi ukuqina. Vala ukusetyenziswa kwezifo hepatic kukho imbali omzimba. Izimo kusetyenziso na unyango Mao inhibitor. Awukwazi ukuthatha iipilisi sixinezelekile, igazi hemolytic, kunye iposi engabalulekanga kwinqanaba nokoyika zophuhliso.
Musa ukumisela amayeza e pheochromocytoma abantwana abangaphantsi kweminyaka emithathu ubudala nangovakalelo eyodwa amacandelo ukwimo iziyobisi.
Ngononophelo kakhulu kufuneka uthatha izigulane iipilisi kunye insufficiency kwezintso. Oku kufuna uhlengahlengiso idosi. Ukuze sibe phantsi kweliso elibukhali likagqirha ngexesha kunyango, izigulane kufuneka diencephalic syndrome, abantu abadala, abantwana ukusuka kwiminyaka emithathu ubudala.
"Dopegit" ngethuba lokukhulelwa zisanyisa
Drug "dopegit" sisetyenziswa ngokubanzi nokubeleka iminyaka engaphezu mahlanu. Ngeli xesha, akukho ziganeko zenzeka kunye neziphumo eteratogenic lwamachiza ekukhuleni kosana olungekazalwa. Ngenxa yokuba ulingo lonyango sele ifakiwe umngcipheko ekude yokuba sesichengeni amacwecwe kwi mbungu.
Ichiza ngexesha lokukhulelwa iwela ngumkhaya, ngoko isigulane kwi 'kwindawo' kufuneka abe phantsi kweliso unyango rhoqo. "Dopegit" ngexesha lokwaphusa (reviews qaphela ukuba oogqirha azilukhuthazi iipilisi usela lwebele-lwebele) ludlulele ubisi lwebele. Ngexesha unyango ugqirha bacetyiswa ukuba ziphazamise nokuncancisa.
Xa bekhulelwe, baqale unyango amayeza veki lamashumi sokukhulelwa. Abantwana abazelwe abafazi abaye baphathwa "Dopegitom" akazange abe naziphi na iingxaki. Into eyahluke yabonwa kwabasetyhini abakhulelweyo abaye benqaba kuthomalaliso le arhente. abantwana bazalwa kunye zizigulo zemithambo eziye zavela ngenxa yokuba ixesha elide oxygen yindlala.
Drug "dopegit" ngexa lokukhulelwa:
- Oku kunciphisa ukuxhathisa semithambo peripheral.
- Kunciphisa ukwenziwa renin.
- Oku kukhokelela kuxinzelelo oluqhelekileyo ukuzala.
- Ngokupheleleyo indawo dopamine - icandelo oku kukhulisa uxinzelelo lwegazi.
- It has a isiphumo kancinane umthomalalisi.
Ngokwezonyango, icikidwa ukuba ichiza banokubenzakalisa umntwana, ungena ngumkhaya okanye ubisi lwebele. "Dopegit" umyalelo ngexesha lokukhulelwa (reviews bathi eli chiza engeyongozi usana) uncoma ukumisela xa inzuzo babenokuba unina kakhulu idlula ingozi usana.
Indlela isicelo, idosi
Medicine "dopegit" lisetyenziswa ngomlomo. Iipilisi nje zingahlafunwa kwaye wahlamba phantsi ngamanzi. Iipilisi Nothabatha esiqingatheni seyure phambi kokuba isidlo okanye imizuzu engama-30 emva kokuba.
Iintsuku zokuqala ezimbini amayeza acetyiswa ukuba asele 0.25 g kathathu ngemini. Umthamo umiselwe isekelwe phezu uxinzelelo lwegazi. Ngonyamezelo elungileyo ithamo ebegqwese qho iintsuku ezimbini. Emva kweentsuku ezintathu zonyango, "Dopegitom" ivela isiphumo ukukhanya uzole.
Izinga izigulana lwegazi ngu 0.5-2 g Oku yahlulwe izabelo ngokulinganayo anigqibele ukuya kane ngemini. Idosi iphezulu ngemihla 3 g
Xa ukufumana idosi yemihla ngemihla unyango 2g lungenasiphumo, yaye ingcinezelo lifinyele embi, i "dopegit" emiselweyo zidityaniswe namanye amachiza umfutho, okanye uyitshintshe ufake enye iziyobisi.
Amayeza elinokunikwa izigulane osebenzisa ngayo unyango namanye amachiza umfutho, kodwa imeko ukususwa wabo kwixesha elizayo. Kule meko, nokunyanga nge-0.5 g ngosuku, ngokuthe ngcembe, ukuba kuyimfuneko, imali zamachiza lande ngamakhefu kweeyure ezingama-48.
abantu abadala kufuneka uqale unyango kunye 0.125-0.25 g Kufuneka uthathe ngaphezulu kwe-2 grams ngemini. Kubantwana ababudala ukususela kwiminyaka emithathu ireyithi emiselweyo amayeza of mg 10 kilogram sobunzima lomntwana ngamnye. Umthamo ngenxa yahlulwe kwizigaba eziliqela.
Musa ukuthatha ngaphezu kwama-65 mg iziyobisi kwekilogram ubunzima bomzimba kunye idosi yemihla ngemihla nganye mayingabi ngaphezu kweminyaka emi-3 Emva kweenyanga ezintathu usebenzisa "Dopegita" lidla kubonakala nokunganyamezelwa ichiza. Kulo mzekelo, womchamo kunye antihypertensives ngakumbi emiselweyo.
"Dopegit" Amayeza: imiyalelo ukuze zisetyenziswe ngexesha lokukhulelwa
Iingcali Ukubuyekezwa uqaphele ukuba la macwecwe zenziwa lula kwaye phantse akukho iziphumo ebezingalindelekanga. Ngenxa yoko, badla kumiselwe kokumitha. Eli chiza Izimo ezimbalwa kwaye akukho iziphumo yityhefu ekukhuleni kosana olungekazalwa. Le ipropati yenza kube lula ukuba ukukhulelwa kwakhe ixesha elide, de ukunikezelwa. Xa bekhulelwe, iipilisi unyango kufuneka ikhatshwe kweliso likagqirha nawazibonayo uvavanyo lwegazi.
Kuthiwa ngokukhawuleza kukhokelela kuxinzelelo oluqhelekileyo "dopegit" ngethuba lokukhulelwa, ncomo. Umthamo uzimisele ngabanye ugqirha. umfazi ahlolwe. Emva koko, ngokusekelwe kwiziphumo wohlalutyo zilungiswe zedosi. Ngokuqhelekileyo eqala unyango kunye enye elucwecweni 250 mg ngosuku. Kubonakala ngathi iziyobisi kunyanyezelwa. Ngonyamezelo mhle ukwandisa ithamo emva kwesithuba seentsuku ezimbini. Ukuthatha ichiza kangangoko nje kwawena zibuyele esiqhelweni. Le idosi iphezulu yemihla ngemihla ukuba abasetyhini abakhulelweyo - 2 Iminyaka
"Dopegit" amanenekazi kwi indawo ayinikiweyo kuphela kwiimeko ezingxamisekileyo kakhulu. Ngokuqhelekileyo, le trimesters wesibini nowesithathu. Ichiza kuyafuneka ukhulelwe ukunqanda yokukhulelwa kade, nokuba ingane iyakhula ngokuqhelekileyo.
Iyeza kunceda ukuze bawubuyise ingcinezelo 10-20%, nto leyo evumela lady okhulelweyo ngokuqhelekileyo uzive.
imiphumela emibi
Tablets "dopegit" ncomo okhulelweyo ingqalelo ichiza ilungileyo ukuzinzisa uxinzelelo lwegazi. Ngaphandle koku, ichiza kunokubangela iziphumo ezingalunganga ezifana ezifana ukozela, silale, ukudideka. Xa ufumana iyeza maxa wambi kuvela ukukhubazeka yobuso, isiyezi, iqinelwa engazinzanga, parkinsonism. Ukusuka ngokuthatha amayeza unobangela yintloko, intolerance lwegazi, myocarditis, bradycardia, ukwanda sisifo sentliziyo kunye angina. Kwakukho nokudumba peripheral, ukuxinana, pericarditis.
In therapy "Dopegitom" wabonakala glossalgia, kome emlonyeni, urhudo, ukugabha reflex, sikabhobhosi. Nomonde iipilisi xa uthatha ungase uphazamise hepatotoxicity, nenyongo, kunye pancreatitis. leukopenia Fixed, agranulocytosis, igazi hemolytic kunye thrombocytopenia.
Eli chiza ingenza myalgia, arthralgia, kunye gynecomastia. Ukumqumbisa galactorrhea, amenorrhea kunye hyperprolactinemia. Nciphisa yobuntu kanye amandla.
Kwiimeko ezinqabe kakhulu, unyango fever yenzekile, Lyell engqondweni. izigulane zabagula ukungxama, angawokubhuda. Bekukho ukuxinana ngeempumlo kunye nokudumba kwamadlala amathe.
ezikhabhathini, indlela yokugcina
Ichiza yenziwa e Hungary ngu "EGIS". Ichiza kufuneka igcinwe kwiqondo lobushushu lwe ukususela +15 ukuya + 25 ° C. Kwindawo wasikhusela ilanga kunye nabantwana. Aphezulu wobomi tablets - kweminyaka emihlanu. Amayeza ayikwazi ingasetyenziswa emva kweli xesha.
Amaxabiso amayeza
Kucetyiswa ngamandla ukuba udibane nogqirha phambi kokuba usebenzise "dopegit" imiyalelo ukulungiselela ukusetyenziswa. Izimvo oogqirha bathi eli yeza aphephe zonke ukunciphisa uxinzelelo, ngoko, oko kumiselwe abafazi abakhulelweyo.
Amayeza zingathengwa phantse yonke ekhemisti. Ixabiso iipilisi 50 250 mg ngeenxa 200-250 engange.
Izimvo oogqirha
Oogqirha ukumisela "dopegit" iipilisi ngexesha lokukhulelwa. Izimvo oogqirha zibonisa ukuba ichiza alunasiphumo kwi entliziyweni. Musa ukusiphikisa imbonakalo tachycardia kwaye akukho ukunciphisa imveliso intliziyo. Ngokutsho kwabo, ichiza kwandisa uxinzelelo lwegazi ngokunciphisa umthamo yokumpompoza kwegazi, kwakunye ngobunzulu izinga kwentliziyo.
Oogqirha ukuvumela ukusebenzisa amayeza ngexa lokukhulelwa, kodwa ziyakhunjuzwa ukuba kufuneka usele oko kuphela kwiimeko engqongqo. Jonga kwi amachiza akhuselekile. Kuthiwa tablets abakwazi ukwenza umonakalo kusana olungekazalwa kwaye zichaphazela lwalo lokukhawulelana nophuhliso. Ichiza ihlala isebenza ngexesha imini, leyo inzuzo eyongezelelweyo kuyo.
Oogqirha bakholelwa eli yeza buthathaka kwaye phantse nabani na ngaphandle abasetyhini abakhulelweyo, kuba akukho emiselweyo.
Medicine "dopegit" ngethuba lokukhulelwa: ncomo
Mhlawumbi omnye amachiza kwemininzi eqhelekileyo ukuba emiselweyo ngexesha ukhulelwe "dopegit". abafazi abakhulelweyo ochaphazelekayo malunga uxinzelelo oluphezulu lwegazi, ndisisela ukuya ekuzalweni. Bathi ukuba kunciphisa xi ngokukhawuleza nangempumelelo. Bonke abo bathabatha ezi pilisi zonwabile isiphumo, wazala abantwana esempilweni. Bakuphawula abanikaziyo ukuba ichiza alunasiphumo kwi Palsy, kodwa koko, ukunceda ukuthintela yokukhulelwa kamva, inegalelo kuphuhliso eziqhelekileyo usana Esibelekweni.
"Dopegit" ngethuba lokukhulelwa kunye nohlaziyo ezimbi kwabangela. Aba bantu babe ukusebenza phantsi ichiza. Bathi ukuba kwandisa uxinzelelo lwegazi kunye nokubi ngenkankulu kunceda. Kungabangela ubuthathaka kunye ukozela. Abanye awuyithandi i ixabiso kunye nento yokuba ichiza kufuneka ngezo ixesha elide.
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