Zempilo, Amalungiselelo
Ichiza "Istenon": ncomo. "Instenon": imiyalelo esetyenziswa kunye analogue
Yintoni na iyeza njenge "Instenon"? Imiyalelo ukusetyenziswa, ixabiso kunye neempawu ichiza ziza kuchazwa kamva.
Ekwakhiweni, imilo, iyeza inkcazelo
ichiza ngasentla kuthengiswa ntoni ifomu? Kuthekani ingxelo le ncomo kubathengi? "Instenon" ifumaneka kwezi fom zilandelayo:
- Amacwecwe ngeenxa and shiny kunye umgangatho ogudileyo isale kwiqokobhe emhlophe. Izinto eziphambili kumafa zazo zezi zilandelayo: hexobendine (hexobendine kwi ekwimo dihydrochloride) kwakunye etofillin kunye etamivan. Ukongeza, ukwakhiwa kwale amayeza ziquka izinto ezongezelelweyo: talc, nemagnesium stearate, starch pregelatinized, umbona starch kunye monohydrate lactose.
- Isisombululo ecacileyo ezingenambala "Instenon" (inaliti) ilungiselelwe nolawulo intramuscular okanye efakwa. nezithako yalo nayo hexobendine (hexobendine ngohlobo a dihydrochloride), kunye etofillin etamivan. Njengoko ngokuba excipients, ngoko ukusebenzisa disodium edetate, amanzi d / u kunye propylene ethers.
Pharmacology
Indlela Yokuphatha njengendlela nokwenza? Yintoni uhlolo lwezonyango ngayo kuthi? "Instenon" - a medicament indibaniselwano leyo iphucula ukutya nobuchopho ejikelezayo.
Ukusebenza ichiza ngenxa iimpawu kwezinto zalo ezisisiseko. Makhe sihlolisise ngokweenkcukacha ezingakumbi.
Esebenzisa ukusebenza kwawo ukuyilwa reticular, etamivan nako ukubuyisela ukusebenza esiqwini umbefu, izakhiwo subcortical kunye neenkqubo ze-uthinte.
Hexobendine iphucula kwaye ibalekisa nokusetyenziswa glucose and O2 ngenxa ukusebenza lemijikelo pentose kunye glycolysis anaerobic. Oku kwenzeka kuphela phantsi kweemeko ioksijini yindlala kunye ischemia xa kakhulu kakuhle oxidative phosphorylation aerobic. Ukukhuthazwa anaerobic zeendawana amandla igcwala yenziwa ukuze babelane yaye Yindibanisela neurotransmitters kunye nokufunyanwa transmission zobuchopho.
Asikwazi ukuba hexobendine ekwaziyo gulwa iindlela (effect) autoregulation yokumpompoza kwegazi (ezesifuba Cerebral), nto leyo enxulumene ngqo kwimpembelelo pyruvate kwaye zincancise (okt iimveliso of glycolysis anaerobic) kwinkqubo receptor ngcanjana kunye arterioles of intracranial.
Yiyiphi indima edlalwe kumalungiselelo etofillin "Instenon"? Imiyalelo, ukubuyekeza baxele ukuba le nto olwenza ukutya engabalulekanga kwaye yandisa imveliso kwentliziyo, nto leyo eyandisa ngakumbi uxinzelelo (CPP) kwiinqanawa kobuchopho. Kulo mzekelo, uxinzelelo lwegazi systemic akatshintshi.
Etofillina sokukhuthaza ukusebenza NA njengoko kuboniswa ukukhuthazwa ephakathi kunye nezinye izakhiwo subcortical, kwakunye nuclei Isiqu kunye namaziko (kubandakanywa FSK enyukliya, embindini ezingummiselo yawo of vasomotor kunye namaziko zemiphunga ye-luvo vagus).
Xa usebenzisa iyeza "Instenon" analogs ezidweliswe apha ngezantsi, kwiimeko trauma cranial kunye nobuchopho (ivaliwe), ukupheliswa kokubetha kobuchopho iphawulwe zizigulo zemithambo, ukufunyanwa isenesazela kumguli okanye ipoti ye-nkqubo yawo.
ubungqina
Yiyiphi imeko kugqalwa iyeza kuyaphumelela? Oko bathi ngale impendulo? "Instenon" kwakubonisa ukuba zisetyenziswe:
- Iimeko post-ngesibetho;
- izifo imvelaphi semithambo zobuchopho, kwakunye utshintsho ezinxulumene kwiminyaka yokuba isigulane;
- kwegazi zaneleyo zokwenza ingqondo engundoqo kunye neziphumo zayo;
- isiyezi, leyo zibangelwa ukuphazamiseka (functional) ingqondo.
Siphelisa ukusetyenziswa
Le medicament "Instenon" (inaliti kunye neefom neziyobisi ngomlomo kufuneka Izimo efanayo) esalelweyo abeke:
- izifo convulsive;
- imo excitation olunamandla;
- iimpawu uxinzelelo oluphezulu lwegazi (intracranial), kubandakanywa ebuhlungu ixesha elide, ukugabha, kunye nokuphazamiseka ebonwayo;
- sokuwa;
- ubuchopho ukopha;
- hypersensitivity ukuya izithako uthetha.
Ne ngenyameko ingqalelo medicament kufuneka isetyenziswe emva kokuba nobetho, kunye emithanjeni stenosis (carotid), kuye kwavela ngenxa yegazi.
Drug "Instenon": imiyalelo yokusebenzisa
Price of ichiza malunga 350-400 engange. kufuneka kusetyenziswe njani na? Kuxhomekeka ebukhulwini kunye nohlobo arhente sifo ngohlobo kwesisombululo ilawulwa intramuscularly okanye yegazi chu. Kule ekuqulunqeni ampoule isetyenziswa amaxesha-1 ukuya kwezi-2 ngosuku.
Kwakhona, lo medicament inokwalathelwa njenge ukuthontsiza ukumnika efakwa. Kulo mzekelo, oku kwakhona emiselweyo 1 ampoule amaxesha 2 ngosuku, kunye ml 250 ka-5% isisombululo zolwelo of levulose.
Xa ekuphuculeni isigulane kuqhubeka ngohlobo lomlomo therapy beziyobisi. Kulo mzekelo, eli cwecwe kuthathwa ngomlomo isixa lamaqhosha 1-2 kathathu ngemini. Idosi iphezulu yemihla ngemihla arhente yi amacwecwe-5. unyango olunjalo ikhutshwa phandle iiveki ezintandathu.
side isenzo
Ngokutsho kweengcali, ichiza "Instenon" kunqabile kubangela ngayo ezibi. Kwezinye iimeko, xa esetyenziswa ngeedosi eziphezulu isigulane bangafumana intloko ebuhlungu, kwakunye noxinzelelo lwegazi ophantsi nokuphuhlisa bomvu apha esikhumbeni.
Overdosing kunye nokusebenzisana
Imiqondiso yokuba libanda, esi sixhobo zezi yintloko, ukugungxula yobuso , kunye tachycardia. Ukuze ukususa ithi ichiza kufuneka ayekiswe, uze uqhube ukusetyenziswa kwayo, kodwa idosi engaphantsi.
Xa isicelo parallel iziyobisi "Instenon" kunye nezenzi zokunciphisa umsebenzi zegazi (kubandakanywa acetylsalicylic acid), ukuze nande isiphumo antiplatelet, ngenxa impembelelo hexobendine.
Xa efumene caffeine ngeedosi phezulu ukunciphisa ukusebenza konwaywa "instenon".
ulwazi oluthile
Yintoni izigulane kufuneka ukuba phambi kokuba uthathe amayeza kuthethwa ngayo? Ngokutsho imiyalelo apha, ngamanye amaxesha kunye efakwa okukhawulezayo "instenon" isigulane lathotywa kakhulu uxinzelelo lwegazi. Kule nkalo, kufuneka ibe ngaphantsi kwe imizuzu emithathu ixesha ukumnika 1 idosi.
Ngexesha unyango ngale arhente ukuba isigulane kufuneka balumke kakhulu xa usebenza ngoomatshini eziyingozi kunye yokuqhuba.
amachiza afanayo kunye nohlaziyo
"Instenon" kungenziwa indawo ngokusebenzisa ezifana "Citoflavin", "Armadin" "Glycine" "Boluses Huato", "Keltikan", "Meksidol", "Cortexin", "Meksiprim", "nucleo CMF Forte", "neurotrophin "" Tryptophan ". Kufuneka kuqatshelwe ukuba la machiza kufuneka ezibonisa zabo kunye neempawu, ngoko ke kufuneka atyumbe liyincutshe onamava kuphela.
Yintoni bathi malunga abathengi amayeza ngoku? Ngokutsho kwiingxelo zazo, ichiza kunqabile inegalelo kuphuhliso naziphi na iingxaki, ngoko ke wabelwe nkqu nabantwana. reception lakhe kakhulu kuphucula igazi ebuchotsheni khipha nezinye iingxaki kunye imithambo yegazi.
Le ethile kuphela kweli chiza ukuziqhelanisa ngokukhawuleza umzimba ukuya ichiza. Kulo mba, sinokuthi ngenkalipho ukuba "Instenon" kutshintshiselwano Foreign isixhobo ayenzelwanga ukusetyenziswa elide.
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