ZempiloUkulungiselela

Isiza esichasayo-"Naklofen": imiyalelo yokusetyenziswa

Ithetha "umyalelo we-Naklofen" ekusebenziseni uchaza isicatshulwa esichaphazelayo soluhlobo olungenalo i-steroidal , olunefuthe elichazwe ngokuba yi - antipyretic ne-analgesic effect. Eli nyanga limiselwe ukuqeda intlungu yesifo semvelaphi eyahlukeneyo kunye nokunyanga iintlobo ezahlukeneyo zezifo ze-rheumatic. Ngexesha elifanayo, isenzo sesilwanyana esichaphazelayo "Naklofen" (umyalelo wokusetyenziswa uqinisekisa) yinto yokuvimbela i-cyclooxygenase kunye nokuphulwa kwe-prostaglandin. Ngaloo ndlela, eli liyeza linciphisa ngokupheleleyo okanye linciphisa kakhulu ubunzima beempawu zokuvuvukala kunye nokunyuka kokunyuka kweentsholongwane kwiintlobo ezahlukeneyo zesistim. Ukongezelela, le nkunkuma engeyi-steroid inikezela ukunciphisa izinga lokushisa komzimba kunye nokuxinwa kwe-prostaglandines kwi- synovial fluid, mucosa esiswini kunye nomchamo.

I-agent ye-anti-inflammatory Naklofen (umyalelo wesicelo uhlala uhlala kwisethi epheleleyo) ngendlela ye-suppositories yama-rectal, i-gel, iipilisi kunye nesisombululo se-injections. Kwindlela yokwakhiwa kwazo zonke iifom ezidweliswe, isithako esisebenzayo sisisimbo esinjenge-diclofenac.

Sebenzisa i-analgesic drug "I-Naklofen" imiyalelo yokusetyenziswa, ingakumbi icebisa ukuba unyango lwezifo ezahlukahlukeneyo zengqungquthela ezivuthayo. Ngokomzekelo, eli arhente lisoloko lichazwe kwi- spondylitis ye-seronegism okanye i-arthritis yabantwana. Esi sidakamizwa esichasayo siboniswa ukuba sisetyenziswe kwi-spondylosis, ukuhlambalaza kunye ne-gout. Abantu abane-arthrosis okanye naziphi naziphi izifo eziphazamisayo zomgudu kunye namalungu axhasa ukuba basebenzisa i-Naklofen ithuluzi. Izigulane ezineliyeza zisiwe kwi-tendonitis, bursitis, synovitis kunye ne-myositis.

Ukongezelela, uluhlu lweenkcukacha ezichanekileyo zokusetyenziswa luquka i-colic ne-renal, intamo, i-back, ihlombe, isisundu okanye isisindo somlenze, i-edema yesisu kunye nokulimala, ukuvuna, ukunweba kweetoni, imisipha kunye nemigqa, i-osteochondrosis yomgudu kunye nokunyameka kwamalungu, ephakanyiswe Imithwalo yemvelo. Ekugqibeleni, le nkunkuma engeyi-steroid imiselwe ngokunyanisekileyo kwi-dysmenorrhea eprayimari neyesekondari kunye nokungenelela kwamazinyo.

Faka isicelo esi sichasayo esichaphazelayo ngokuchanekileyo ngokungqinelanayo nxamnye nokusetyenzwa kwe-diclofenac, kunye nokukhathazeka okwandisiweyo kwesigulane kwi-salicylates okanye nayiphi na into evela kwiqela le-NSAID. Abantu abanesilonda sesisu esiswini okanye isilonda se-peptic ye-duodenum kufuneka banqabe ukuthatha uNablofen. Iingxelo zikhankanya kunye nokungafuneki kokusetyenziswa kwayo ekuphumeni kwamathumbu emathumbu. Ukongezelela, musa ukumisela lesi sigulo sokuchasana nezigulane ezingaphantsi kweminyaka eli-14.

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