Zempilo, Amalungiselelo
"Kaffetin" (tablets): imiyalelo ukusetyenziswa, analogs, ncomo
Eli nqaku sijolise ichiza elibizwa "Kaffetin". Le Ezipilisi uluhlu lweziphumo, eziquka:
- psychostimulant;
- zokuphelisa iintlungu;
- antipyretic;
- antitussive;
- anti-ukudumba.
Amaninzi isetyenziselwa yintloko. Njengazo zonke amayeza, i "Kaffetina" kukho izikhokelo kunye Izimo, iziphumo ebezingalindelekanga kunye zimpawu kunye nemithi ethile. Konke oku bafunda ngokufunda eli nqaku. Ukongeza, kufuneka ukwazi yaye "Kaffetin" yaye "Kaffetin kukhanya" (eza kuxutyushwa kweli nqaku) zahluke kancinane kumafa. Owokuqala iqulathe codeine, kwaye eyesibini - akukho.
Isakhiwo kunye Nokuhlanganiselwa
Kweli candelo, uza kufunda ntoni "Kaffetin" (cwecwe, ifom ukukhululwa). Okokuqala, hlolisisa ukwakhiwa, kuya kuba lula ngakumbi ukuthatha ngokohlobo itafile. Le kumhlathi osekhohlo iqulethe iziyobisi, kwaye ngasekunene - umxholo yabo milligrams.
paracetamol | 250 |
propyphenazone | 210 |
caffeine | 50 |
Codeine phosphate sesquihydrate | 10 |
glyceryl dibehenate | 6.3 |
Calcium hydrogenphosphate dihydrate | 21.1 |
sodium carboxymethyl starch | 14.5 |
dust Colloidal anhydrous | 2.5 |
sodium croscarmellose | 9.6 |
wemagniziyam stearate | 13.5 |
sodium lauryl sulfate | 1.5 |
povidone | 12.5 |
microcellulose | 28.5 |
Xa uthenga, anikele ingqalelo kumqulu ukuba yonakele, ngoko sebenzisa ichiza angafanele ngayo. Apha ukuze kutshekishwe iipilisi kwi ngokuphuma, anikele ingqalelo ileyibhile, umbala kunye nenani iipilisi xa isitya. Baya kufuneka ikhangeleke ngolu hlobo:
- iflethi, ngeenxa zonke;
- umbala - ezimhlophe;
- umbhalo - «5», Caffetin;
- kwinqakwana namnye oya iipilisi ezintandathu okanye ishumi;
- e ibhokisi iqulethe strip omnye ngaphandle kokuba amacwecwe ezilishumi, okanye ezimbini, ukuba babe tablets ezintandathu.
pharmacodynamics
"Kaffetin" (tablets), ekuthethwe ngayo kweli nqaku, njengoko waba ngokucacileyo, sisiyobisi udibaniso. Icandelo ngalinye ezisebenza umsebenzi ethile. I-paracetamol na le manyathelo alandelayo:
- antipyretic;
- ntlungu.
Caffeine, inxalenye ichiza, uyakwazi:
- ukukhuthaza ukusebenza kwengqondo;
- nokukhuthaza ifuthe iintlungu of paracetamol;
- ukunciphisa ukozela;
- ukususa nokudinwa;
- ukwandisa ukusebenza;
- izinga intliziyo ukwanda;
- nehigh blood.
Codeine unako ukuhlangula khohlo. Oku kwenzeka ngenxa kwezithandani iziko ukhohlokhohlo excitability neuronal kwinkqubo luvo. Kanye njengokuba acetaminophen, codeine, kukho into iintlungu uyakwazi ukutshintsha imbono ngokweemvakalelo intlungu.
Le theyibhile ingezantsi into ebizwa propyphenazone kunceda ephelisa intlungu nokunciphisa lobushushu emzimbeni. ukusebenza iintlungu kwenzeka kwisithuba seyure emva ezithatha ichiza, kodwa kuthatha malunga neeyure ezisibhozo.
Pharmacokinetics
"Kaffetin" Ngoku siza kuxoxa pharmacokinetics beziyobisi. Iipilisi ziyinxalenye paracetamol eziqhelekileyo, nto leyo ako ngephanyazo. Ayithandi eliphezulu kwi igazi ambona kwemizuzu engama-30 emva kokuba yolawulo. Nethe kungenziwa esibindini ngeendlela ezintathu:
- conjugation ne glucuronide;
- conjugation ne sulfate;
- igcwala.
Idubule emva kweeyure ezine nge izintso ngohlobo kwezinto metabolic.
Le peculiarity caffeine kukuba ifunxwe emathunjini onke amasebe. Lula enqumla iplacenta. caffeine obukhulu egazini waphawula emva kweyure 1 emva ulawulo iziyobisi. Le into abelwa ngokukhawuleza kakhulu kuyo umzimba womntu. Caffeine umzimba esibindini mazwe nge izintso emva kweeyure ezintlanu ezinesiqingatha.
Ingakumbi ukufakwa rapid yahlukile, kunye codeine. Xa plasma eyavela eliphezulu ekufikelelwe kuso emva iiyure ezi-2 emva kokuba yolawulo. Lithathwe into nge nezintso, enyongweni unakho uphume ngokusebenzisa iyure 4.
into propyphenazone ifunxwe lokugaya. Egazini, oko kubonakele nemizuzu engama-50 emva kokuba yolawulo. Kwazona kwi enyongweni okanye umchamo kwisithuba seeyure ezimbini.
ubungqina
Kweli candelo uyakwazi ukufumana phandle ngoko ke zibonisa ukuba ukusetyenziswa "Kaffetin ukukhanya" iziyobisi. Imiyalelo yokusebenzisa (tablets) umisela ukuba i-arhente ukuze kuthathwa izifo ezithile kunye ubuhlungu, ezizezi:
- intloko ebuhlungu;
- lizinyo;
- migraine;
- neuralgia;
- myalgia;
- intlungu post-traumatic;
- arthralgia;
- algomenorrhea.
Le izinto ezibonisa ukuba ichiza "Kaffetin" ziyafana. Kuyimfuneko ukuba uyithathele ingqalelo into yokuba imveliso iqulethe caffeine, nto leyo eyandisa umsebenzi ngokwasemzimbeni nangokwasengqondweni. Oko akukhuthazwa ukuba zisetyenziswe phambi lokulala. Thatha ipilisi "Koffetina" kunokwenzeka kwiimeko apho iintlungu kubonakaliswa ngokulinganisela. Intlungu ingaba ngokupheleleyo nayiphi na umthombo.
Izimo
Njengazo zonke amayeza, Izimo zabo kwaye "Kaffetin" iipilisi. Imiyalelo yokusebenzisa beziyobisi ithi ukuba kwiimeko ezithile ezingqalileyo, ichiza kufuneka ingasetyenziswa. Kweli candelo siza kukhangela contraindication ukuya ichiza. Ezi ziquka:
- hypersensitivity;
- ukusilela hepatic;
- ukusilela kwezintso;
- leukopenia;
- ukopha yokudla;
- ukuphazamiseka ixhala;
- izifo nemithambo yegazi;
- zokulala;
- nokukhulelwa;
- zisanyisa;
- kweminyaka elishumi elinesibhozo.
Amatyala ngasentla zithintelwe ngokungqongqo ekuthatheni eli chiza. kuba abantu abasemngciphekweni, zezi:
- Ndaziva intlungu elibukhali esiswini kwaye musa ukuba ityala layo;
- uphethwe somoya;
- babe nesifo semiphunga ezingapheliyo;
- ngubani kwenzeke amahlaba;
- ukuba ukuxhomekeka iziyobisi;
- ubunzima yokusela;
- owandisa excitability;
- kohlobo load;
- ukwaluphala.
Kule meko, phambi kokuba ezithatha ichiza kufuneka kusoloko ubonane nogqirha.
effect side
Tablets "Kaffetin ukukhanya" ngokuthi "Kaffetin", kwaye inokuba neziphumo ebezingalindelekanga. Khumbula ukuba zonke iziyobisi kufuneka zisetyenziswe ngqo ngokwemiyalelo, leyo kwibhokisi kunye ichiza. Musa self-medicate, phambi kokuthatha amacebo kwiingcali. Nkqu amayeza kakhulu kwezinye kunokuba yingozi ukuba ezona imithetho ngokuphathelele ukusetyenziswa kwazo. Ngoko ke, ukuba kwicala ifuthe "Kaffetin" iziyobisi ziquka:
- ucaphuka;
- lafa;
- ukukhathazeka;
- ugwayi;
- ukukhawulezisa kwezinga intliziyo;
- kongeza uxinzelelo;
- ukuqhubela phambili izilonda;
- isicaphucaphu;
- ukuphalaza;
- ufunga kwesikhumba;
- ezindlwini;
- ukulunywa;
- iindumbisa ebusweni;
- bronchospasm;
- nokudumba laryngeal.
Mhlawumbi kungenzeka kunye okanye ngokwahlukeneyo. iziphumo ebezingalindelekanga zinqabile. Ukuba naziphi na iimpawu zezi kwaba, kufuneka uqiniseke ukuba wazise ugqirha wakho. Uya kukuxelela indlela ukujongana nengxaki, mhlawumbi ucebise ichiza olufanelekileyo ngakumbi.
"Kaffetin": imiyalelo yokusebenzisa
Tablets "Kaffetina", njengawo onke amanye amachiza kufuneka zisetyenziswe ngqo ngokwemiyalelo, ukuze abangele libanda, iziyobisi. Le idosi iphezulu yemihla ngemihla - tablets ezintandathu.
Ubude unyango kufuneka ingadluli kwiintsuku ezintlanu. Noko ke, ugqirha kunokwandisa idosi yemihla ngemihla ikhondo unyango. Ngaphandle isindululo ngugqirha wakhe, la manyathelo kungenziwa.
libanda
Ngokusisiseko, thatha ezi pilisi ukuba intloko ebuhlungu. "Kaffetin" kufuneka basela ngqo ngokwemiyalelo. Icandelo ngalinye libanda, lubonakala ngeendlela ezahlukeneyo. Ukuba Ladlula izinga paracetamol, ngoko mpawu zilandelayo:
- isikhumba kuba luthuthu;
- isicaphucaphu;
- ukuphalaza;
- umsebenzi kwesibindi kakuhle.
Oku kwenzeka emva kweentsuku emva nomthamo. Ukuba ngaphezu ithamo caffeine:
- bekhathazekile;
- lafa;
- intloko ebuhlungu;
- ukudideka.
Ukuba udlule umthamo codeine, kuvela ezi mpawu zilandelayo:
- xhopho ebandayo clammy;
- nesiyezi;
- ukozela;
- zokucutha;
- uvalo;
- nokudinwa;
- yobuthathaka;
- ukuphelelwa umoya;
- ukukhathazeka;
- yombono.
Ukuba uqaphela iimpawu ze-libanda, ngoko kukho imfuno engxamisekileyo ubize inqwelo yezigulana. Musa ukuzama iphume isisu kuphela. Oku akwanelanga, kuyimfuneko ukuba ukubuyisela intliziyo wegazi.
"Kaffetin Forte" macwecwe: baphendule
Imiyalelo ukuba eli chiza kuthiwa "Kaffetin" kufuneka zisetyenziswe kunye amayeza zilandelayo:
- barbiturates;
- iziyobisi ukuze sokuwa;
- rifampicin;
- zidovudine;
- ethanol.
Okhankanywe ngaphambili, ukuba le mveliso ziquka paracetamol, oko kunceda ukuqinisekisa ukuba ukupheliswa ngokupheleleyo konyuso chloramphenicol ngokuphindwe kahlanu. Ubukho caffeine kukhokelela nokufunxwa kakuhle ezinye izinto. A codeine kuphucula iziphumo analgesics kunye ipilisi zokulala.
Ukuthengiswa, ukugcinwa, ixabiso kunye nemiyalelo ezizodwa
Eli chiza ekhululwa kwikhemesti kuba ngqongqo kagqirha. Gcina "Kaffetin" imi kwindawo emnyama, kude ebantwaneni. Iqondo lobushushu Igumbi kufuneka ingadluli 25 degrees Celsius, kwaye ibe ngaphantsi kwe 15. lokugcinwa kwezinto ichiza yiminyaka emithathu.
Xa ekufumaneni ichiza kufuneka kululahla ukusetyenziswa kotywala. "Kaffetin" uyakwazi ukuzigqwetha kancinci iziphumo zovavanyo. Iimbaleki kufuneka bazi ukuba ichiza liyitshintshe iziphumo ulawulo nokusetyenziswa kweziyobisi. Ixabiso indlela nama-115 engange.
Nokubuyekezwa analogue
"Kaffetin" - iipilisi ezinceda ukuphelisa intlungu. Analogue zezi:
- "Paracetamol" (18 engange).
- "Trigan-D" (70 engange).
- "Solpadein" (140 engange).
Izimvo yale ukulungiselela esihle kakhulu. Kukho iimeko nekunqabileyo nesiyezi kunye isicaphucaphu.
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