Zempilo, Amalungiselelo
"Lomfloks": imiyalelo ukusetyenziswa, ixabiso, analogs
Kutheni iziyobisi ezifana "Lomfloks" linokukwenziwa? Imiyalelo ukusetyenziswa, Izimo nokubonakaliswa ngenxa yokwamkela ichiza ziya kuqhutywa ngokweenkcukacha kweli nqaku. Ukongeza, uya ufunde eli chiza kuyo iyafumaneka, zeziphi izinto ziyingxenye kuyo, loo nto ikutya kwaye nokuba yena analogs naluphi na uhlobo kangakanani.
Iipakethe ichiza, zayo imilo, inkcazo kunye nokwakheka
Ziziphi fom isiyobisi loo ndawo ngokuthi "Lomfloks"? Imiyalelo yokusebenzisa yazisa ukuba medicament esebenzayo yenziwe kuthengiswa kuphela ngohlobo amacwecwe camera (film) amacwecwe lume (400 mg) njenge umbala ukukhanya omdaka.
Icandelo esebenzayo yale kwiarhente lomefloxacin (Zisebenziselwa hydrochloride). Ngokuphathelele amacandelo ezongezelelweyo, ngoko ke ziquka lactose, talc nyulu, starch, crospovidone, polyvinylpyrrolidone, isodiyam lauryl sulfate, propylene ethers, nemagnesium stearate, sodium starch glycolate kunye colloidal lesilicon dioxide.
Ukubunjwa yeqokobhe enokukhokelela izinto zilandelayo: chloride methylene, isopropanol, titanium dioxide kunye hydroxypropyl methylcellulose.
"Lomfloks" ezi amacwecwe namadyungudyungu (iziqwenga 5) zibekwe zibe kwiibhokisi kwikhadibhodi.
Njengoko imisebenzi iziyobisi?
Yintoni na ichiza "Lomfloks"? Imiyalelo yokusebenzisa icebisa ukuba le arhente i arhente zokwenziwa elwa. Lingcwaba lomfo iqela fluoroquinolone amayeza kwaye spectrum ezibanzi amanyathelo bactericidal.
Izincomo ikwazi ichiza le ethintela iibhaktheriya DNA gyrase, ngaloo ndlela bakha tetramer kunye entsokothileyo kwaye ukuphazamisa ukuphindaphindeka nokubhalwa DNA. Ngenxa yokuba sesichengeni ezinjalo kukho nokutshatyalaliswa iiseli izifo.
Le medicament iyasebenza nxamnye gram Cya ezingakhiyo, kunye Igram HIV kunye aerobes. Ngaphezu koko, ichiza kungaba yingozi chlamydia, Mycobacterium tuberculosis (imi obuvakalayo extracellularly), kwakunye ezinye strains uroplazmy kunye mycoplasma.
Kwimeko-bume asidi ukusebenza ichiza lifinyele kakhulu, kunye nokumelana kuphuhlisa ngokucothayo kakhulu.
Eli chiza kunempembelelo postantibioticski ngokukhawuleza.
Kufuneka kwakhona uqaphele ukuba streptococci kunye anaerobes abanganyangekiyo yesenzo lomefloxacin.
Pharmacokinetics
amayeza wona aya Ugxile nini "Lomfloks" (tablets)? isicelo Umsebenzisi ithi emva ulawulo kwi icandelo layo esebenzayo ako phantse ngokupheleleyo ukusuka lokugaya.
Ngokusebenzisa 400 mg le kuqulunqo ingqalelo yayo ephezulu egazini waphawula emva kweeyure 1.5-2 kwaye imalunga 3,2-5,2 mg ilitha nganye. Kufuneka kuqatshelwe ukuba xa ufumana medicament in wathi umthamo lomefloxacin lamanani ukuze igqithe MIC lwegciwane ezininzi. Ubuncinane ngenxa isiqingatha imini.
Unxibelelwano into esebenzayo kwiiproteni plasma bamalunga nama-10%. Lomefloksatsin ngokukhawuleza ingena kuzo zonke izihlunu zomzimba. Uyondelelwano lwee- kweziyobisi kwiincindi ababazalayo amaxesha 3-6 ngaphezulu kwi-plasma, ingakumbi kwizihlunu yesinye, macrophage kwemiphunga kunye nomchamo.
Isiqingatha umphefumlo element esebenzayo nama-7-9 iiyure. Malunga nama-70-80% of lomefloxacin na imveliso emini (ekwimo unmodified) kwi yokuchama.
Xa izigulane umsebenzi othile kidney isiqingatha-ebomini element esebenzayo inyuswe kakhulu.
ubungqina
Zeziphi izifo prescribers "Lomfloks"? Imiyalelo yokusebenzisa iqulethe ezi okukhomba zilandelayo:
- izifo ezihlasela zosulele ngokuphefumla (ezosulelayo), okanye kunoko, amaqela ephantsi (kubandakanywa exacerbation yomoya ezingapheliyo kunye pneumonia);
- Izifo ezosulelayo kunye ukudumba eziye zabangelwa iintsholongwane ezibuthathaka ukuba lomefloxacin;
- media otitis;
- lwechlamydial ezingapheliyo kunye etsolo, usuleleko gonococcal exutyiweyo;
- izifo enzima lula le wokuchama kunye neenkqubo zokuzala;
- Izifo ezosulelayo izicwili ezithambileyo kunye nesikhumba;
- cholecystitis kunye enterocolitis esosulelayo;
- izifo amalungu kunye namathambo, kubandakanywa osteomyelitis ezingapheliyo;
- nesifo sephepha yemiphunga (kubandakanywa iindlela zosulele phambili zesi sifo, iintsholongwane drug resistant, ukunyamezelana rifampicin, isifo sephepha ezihamba iinkqubo nonspecific arhabaxa).
Kwakhona qaphela ukuba ichiza ingqalelo rhoqo ezimiselweyo nokuthintela iingxaki ezosulelayo kwiinkqubo utyando transurethral.
Izimo
Ukuba kukho ukungaqheleki kuyo nayiphi na imeko asikwazi ukuthatha iipilisi 'Lomfloks "? Imiyalelo zokusetyenziswa (ixabiso ichiza ziyachazwa ngezantsi) iqulathe uluhlu zilandelayo Izimo:
- ngexesha yokumitha nokuncancisa;
- sokuwa, yegazi ebuchotsheni, kwakunye kurhulumente, ehamba yombono;
- Abantwana ukuya kutsho kwiminyaka engama-15;
- hypersensitivity nomonde ukuba lomefloxacin nezinye quinolones.
Medicament "Lomfloks": imiyalelo yokusebenzisa
Inkcazelo yale sixhobo usoloko efumaneka imiyalelo apha. Ukongeza, ukuvula ukuba ichiza ulwazi izigulane malunga ulapha Kufuneka ikhutshwe kwi unxaxho elinikiweyo.
Tablets "Lomfloks" kufuneka lincance (amanzi othululwayo kubushushu room). ukusebenza kwayo akuxhomekekanga ekudleni. Umthamo eqhelekileyo kule kuqulunqo yi mg 400 kanye ngemini.
Xa kakuhle umsebenzi kwezintso ngosuku lokuqala unyango emiselweyo 400 mg iziyobisi, kwaye elandelayo - 200 mg (kanye ngosuku). Le idosi ixesha unyango zixhomekeke ebukhulwini ecaleni kunye susceptibility ezikhoyo.
Kwimeko apho umntu ene-iipilisi TB "Lomfloks" kufuneka zidityaniswe kunye iziyobisi ezifana "isoniazid", "pyrazinamide" yaye "Ethambutol".
Ngelo xesha linye ayinqweneleki kakhulu ukuthatha lomefloxacin ne rifampicin. Oku kungenxa yokuba ezi izinto ezi abamelene kukhuphiswano.
Ingozi abasabela nomsi kube kakhulu kuncitshiswa ngokuthatha Lomfloks iipilisi ' "ngokuhlwa.
imithi
Xana ndzi nga wu namanye amayeza amayeza "Lomfloks"? Imiyalelo yokusebenzisa (esebenzisa analogue ziya kwenziwa ekupheleni nqaku) uthi ukuba ichiza uyakwazi ukwandisa umsebenzi anticoagulants zomlomo, kwakunye ukwandisa ubuthi NSAIDs.
Asidi kunye sucralfate yokufunxa kade beziyobisi kunye nokunciphisa bioavailability yayo, kusekwe inamehlo chelate. Ngokumalunga ulwamkelo ngaxeshanye kunye probenecid, usenza inhibition of zinomgutyulo kwezintso.
imiphumela emibi
Ikha nefuthe elibi emzimbeni iziyobisi womntu "Lomfloks"? Imiyalelo yokusebenzisa (ncomo, analogs thaca kweli nqaku) ithi arhente eyaziswa unawo iziphumo ebezingalindelekanga kulandelayo:
- Imikhumbi nentliziyo: Vasculitis kunye nengcinezelo ukusebenza kwenkqubo Cardio-miphungeni.
- isixokelelwano sokuphefumla: nokudumba kwemiphunga kunye kwingqula.
- Umzimba: komzimba reactions, photosensitivity, anaphylaxis kunye angioedema.
- Kokudla: ukudumba okwenziwa sisilonda pseudomembranous efakwe ngayo isifo ngomlomo.
- Isibindi: uphuhliso kwesibindi.
- Ochama: polyuria, nephritis Embi, ukugcinwa wokuchama kunye ukusilela kwezintso.
- Izihlunu / skeleton: tendonitis, komsipha lungu, arthralgia kunye myalgia.
- I-luvo (neuropathy kunye central): ixhala, Ataxia, ukudideka, unditsho, ukudakumba, iingcangcazela, zokulala, isiyezi, ukuphazamiseka kwengqondo, intloko ebuhlungu, ukuba nemibono, ukungaboni, incasa enxamnye, photophobia kunye diplopia.
- Yesikhumba: hyperpigmentation, dermatitis exfoliative, Stevens-Johnson syndrome kunye epidermal necrolysis.
- Nethe: Hypoglycemia.
- Igazi: igazi haemolytic kunye thrombocytopenia.
oyi
Zeziphi iinkalo machiza kufuneka bazazi izigulane, phambi kokuba bathathe "Lomfloks" tablet? Inkcazelo yokulungiselela, imfundiso efunekayo ukufunda, kwakunye thethwano zokuqala yincutshe.
Xa isifo enjalo, njengoko kwesibindi,-hlengiso nomthamo irejimeni kuyimfuneko. Kodwa kuphela xa umsebenzi izintso ukuba ivuke.
Ngexesha unyango, iyeza kuyimfuneko ukuphepha utyhileko UV eyingozi.
Asidi, kunye neevithamini, kunye nezinye ii-arhente eziqulathe aluminiyam, nemagnesium nesinyithi, kufuneka kuthathwe kwiiyure ezimbini ngaphambi kunye iiyure ezimbini emva kokuba ezithatha ichiza phantsi ingqalelo.
Ngaba uyakwazi ukuqhuba isithuthi kunye nolawulo amayeza ngu iindlela ezahlukeneyo, "Lomfloks"? Imiyalelo zokusetyenziswa (ixabiso le mveliso idweliswe kwicandelo ngezantsi) yazisa ukuba esi sixhobo kungabangela ingqalelo nkene kakhulu Uyagula. Kulo mba, kungenzeka izinto eziyingozi kufuneka isigqibo kuphela emva kokuba kwenziwe uvavanyo impendulo yesigulane namayeza.
Analogs "Lomfloks" ncomo ixabiso iziyobisi
malunga nokusetyenziswa kwemali sikhokelo ingxelo ziye zabonakaliswa kweli nqaku (ukulungiselela iinjongo zemfundo). Njengoko ngexabiso, kunokwenzeka ukuba ukwazi iindleko ngqo kuphela ezikhemisti. Ngokuqhelekileyo, i-avareji yahluka phakathi engange 500 (tablets 5).
Yintoni enye ukuze kuthi ngalo ichiza imiyalelo 'Lomfloks "ukusetyenziswa? Analogue beziyobisi ndamgqala ngokweenkcukacha. Ngokutsho kwakhe, lo iyeza kutshintshwa yimithi zilandelayo: ". Lomefloxacin hydrochloride" "Ksenakvin", "Okatsin", "Lomatsin", "maksakvin", "lomefloxacin", "Lofoks",
Njengoko ngokuba ujongo, ukuba elincumisayo becala. Izigulane bathi "Lomfloks" ipilisi kakhulu ngempumelelo ulwe usulelo. Nakuba kunjalo, kufanele kuqatshelwe ukuba abanye abantu olu nyango rhoqo akhalaze yeziphumo ebezingalindelekanga.
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