Zempilo, Ukulungiselela
"Olanzapine": iifanekiso, inkcazo yokulungiselela, imiyalelo yokusetyenziswa
Kuba unyango ngesifo kunye disorder amachiza ukusetyenziswa ngokusekelwe olanzapine kweziyobisi. Kukho iziyobisi ezininzi amagama zorhwebo ezahlukeneyo, kodwa isiphumo esifanayo antipsychotic. Enye isiyobisi okunjalo iziyobisi "olanzapine" analogs ziqulathe kumafa yayo eyona nto iyonke esebenzayo.
Inkcazelo yokulungiselela
Oku kwenziwa yi-arhente antipsychotic "ALSI Pharma" ZAO njenge amacwecwe umbala otyheli, imilo leyo ufana biconvex njengesilinda.
Ubume ichiza zakha izithako engasebenziyo, eziquka uhlobo microcrystalline kwincindi, monohydrate lactose, lokufaka krospovidonovy, wemagniziyam stearate. Inani labo kwandisa kumaxesha ezimbini, ezintathu okanye ezine, ngokuxhomekeke olanzapinovoy balawule.
Amacwecwe afakwa ezingxobeni zonke lidle ngamaqhekeza 7 namadyungudyungu kwi umqulu oluno iziqwenga 4 okanye 8.
Lithetha "olanzapine" Umsebenzisi Isicelo inxulumene amachiza antipsychotic neuroleptic leyo kombisa noFaro ngenxa serotonin, dopamine, muscarinic, adrenergic kunye histamine receptor Ukwakheka.
Emane kunciphise umsebenzi excitatory ye-luvo dopaminergic mesolimbic, Umsebenzi kancinane Uhanjiso luvo striatal, elawula ukusebenza injini. Ukwehla amandla kwi ikhaliphe eqhelekileyo yokhuselo, ukuba usebenzisa i idosi eliphantsi ngaphandle ebangela ebuthongweni cataleptic.
Medicine "Olanzapine" kwandisa ukusebenza anxiolytic lomsebenzi test "anxiolytic" ngoxa ibaleka. Ithwala uyeka nezingalunganga enemveliso njengoko iimfeketho zokufeketha nemibono hallucinatory.
Into esetyenzisiweyo
Tablets "olanzapine" isiphumo bafakela imeko seSkitsofreniya ebudaleni kwinqanaba etsolo, njengokuba ukugcinwa kunye nonyango protivopovtornogo elide. Bona zisetyenziselwa disorder ngengqondo kunye iimpawu evuzayo iimfeketho zokufeketha, imibono hallucinatory kunye neempawu ezimbi ezifana flattening ngokweemvakalelo, ukunciphisa imisebenzi ebalulekileyo ekuhlaleni, zokuncipha apparatus kwezwi.
Drug bayiyeka ukuphinda uxhuzula kunye eguquguqukayo, ukuba cwecwe aphathe ngempumelelo izigaba manic.
Ukulungiselela "olanzapine" kukhutshwa abadala kunye nezigulo bipolar Uthando ngohlobo monotherapy okanye kubanjiswene imithi equlathe ion lithium okanye valproic acid. Ichiza isetyenziselwa ukunyanga iifom zosulele manic okanye oxutyiweyo yezenzo ezingenzeka iimpawu zengqondo, kwakunye sibe manqanaba utshintsho ukuzila.
Lithetha kudityaniswe amayeza fluoxetine ukuba iimeko edakumbisayo ezihlobene ne kwengqondo.
Imiqathango yosetyenziso
Medicine yesicelo "olanzapine" Umsebenzisi icebisa imini 0,005 ukuya 0,02 g ngomlomo ngaphandle unamathele imo amandla.
isimo seSkitsofreniya izigulane abadala aphathwe kunye idosi yokuqala mihla le 0,010 g
mania etsolo abadala, ukuphazamiseka ngokweemvakalelo luphawulwa, isuswe yonke imihla mabaphakelwe olanzapine in 0.015 g lulungiselelwayo kanye. Ukuba amacwecwe zisetyenziselwa ifuthe ukugcinwa kunye amayeza esekelwe Lithium ion okanye valproic acid, ngoko yaphathwa idosi yemihla ngemihla ka-0,010 g ngalinye kanye.
iinkqubo depressive ebudaleni disorder ngenxa eguquguqukayo, sizani yonke imihla mabaphakelwe 0,005 g, kudityaniswe fluoksetinovogo kweziyobisi 0,020 g. Ukuba kukho imfuneko, ngoko ukuba hlengiso wemithi amayeza.
Kuba izigulane abadala kunye nesisongelo kunokwenzeka kakhulu insufficiency kwezintso okanye sesibindi njengaxa kukho imingcipheko enxulumene nesini nemazi, saka ubudala-xa olanzapine deceleration exchange imali yayo ekuqaleni ngemihla kuyehla 0,005 g
ezi zixhobo
Medicament "Olanzapine" isasetyenziswa uye amagama zorhwebo ezahlukeneyo. Bona liveliswa abenzi basekhaya angaphandle.
Phakathi kubavelisi Russian ukujikeleza-off iinkampani 'iziyobisi Technologies "kunye ichiza" Olanzapine-TL ", azipilisi 0,0025 g umboniso camera.
Amanye amayeza zasekhaya yindlela "Olanzapine", yenziwa yi-JSC "North Star". Kukho elucwecweni kunye ukutyabeka ifilim kunye ne nedosi ye-0,005 g
mveliso Russian "Kanonfarma lweMveliso" JSC wavelisa ichiza "Canon of olanzapine."
amayeza Israeli liyeza "Olanzapine Teva," iinkampani imveliso "Teva Pharmaceutical Enterprise Co., Ltd.".
Togu Slovenian kusho "Zalasta Cu tab", emacwecweni 0,015 g ukuya resorption. Eyenziwe kwishishini "Krka, Novo mesto." Kwakhona data eziveliswa "Zalasta" Amacwecwe iziyobisi.
Swiss analogu ichiza njenge "Zyprexa" njenge lyophilisate kwi ezineengqayi, ukusuka apho isisombululo silungiselwe ulawulo intramuscular, ne nedosi ye-0,010 azipilisi esasazekayo 0.005 grams ikhona iziyobisi "Zyprexa Zidis". Bona eveliswe yi "Eli Lilly Vostok SA". Kwimarike zamayeza kukho "Zyprexa Afrika United" medicament olungumgubo akusebenzi 0,21 g
inkampani Polish "Polpharma" amayeza eyenziweyo "Normiton" iipilisi kunye ukutyabeka lisesingxobeni ka 0.005 g
Drug "Olanzapine" isasetyenziswa Hungarian eziveliswa "kaGidiyon Richter" ngokuba macwecwe "Parnasan" kwaye zoxubo mayeza zezityalo "EGIS" iziyobisi kuphuhliswa "Egolanza".
Inkcazelo "Zalasta" iziyobisi
Oku kubhekiselele neuroleptic antipsychotic. macwecwe Ukukhanya yellow ezingeenxa, imilo biconvex kancinane kunye namabala amnyama. Kukho ezintandathu iidosi: 0,0025 g, 0,005 g, 0,01 g, 0,015 g kunye 0,02 g olanzapine. Awongeziweyo amaqela ingqalelo Cellactose opholileyo, starch pregelatinized nengqolowa ifomu, amanzi emzimbeni aerosilovy Yinxalenye, wemagniziyam stearate.
Uphawu azipilisi "Zalasta" yemiyalezo ichaza nobhalo ngohlobo lwe nemikrolo inkcazo idosi. iiphakheji nomthengi ipleyiti ulinywa iipilisi 7. Umqulu inokuba liqulathe 4 okanye 8 of kumadyunguza ezinjalo.
Le arhente neuroleptic ebonisa imisebenzi ebanzi imithi. ukusebenza Antipsychotic ezinxulumene uhlobo mayiqhagamshelane iimanyano dopamine receptor. umsebenzi okulalisa zibangelwa elekhtrons sites adrenoceptor ukuba zenza ukusekwa reticular kwi kwiiseli ze stem ebuchotsheni.
umsebenzi Antiemetic kunokwenzeka kwi stop D 2 receptor -dopaminovogo aninasabelo kwindawo aqala-uhlobo leyo ifumaneka kwiziko emetic.
indima Hypothermic ikhutshwa phandle ngokubhloka ilitye le dopamine receptor lweentlobo kule ngxenye.
Medicine "Zalasta" yemiyalezo icebisa esebenzisa ekubonakalisweni seSkitsofreniya. Iipilisi bayakwazi ukuba sihlale sixakekile abacombululi iimpawu zonyango ngexesha kunyango ixesha elide kwezigulane ukususela ekuqaleni emihle ichiza.
Kuthethwa ukuphelisa mania episodic ngendlela oluphakathi okanye ezintsonkothileyo. Iipilisi nokuziphatha isilumkiso ngokulungisa uphindaphindo phithi bipolar kubantu abane ngeziqendu manic.
Ichiza ilungiselelwe ulawulo yomlomo kanye ngemini. Amasuntswana ukutya zingakuchaphazeli inkqubo ukufunxeka olanzapine, leyo ikuvumela ukuba usebenzise cwecwe ngalo naliphi na ixesha. Phezu kurhoxiswe ichiza ngokuthe ngcembe ukuba sinciphise idosi.
Kuba unyango ukuphazamiseka seSkitsofreniya lisetyenziswa nomthamo yokuqala ka-0,010 grams ngemini.
Iziqephu mania baqalisa aphathwe idosi yemihla ngemihla ka-0.015 g lulungiselelwayo kwisicelo elinye okanye 0,010 grams xa zidibene nezinye neuroleptics.
uthintelo phindwa disorder kwi eziphango inyathelo oluqhutywa primary beleni medicament 0,010 grams ngemini. Ukuba abantu bathatha isixhobo ekulungiseni mania episodic, ekuya kuqhutyelwa unyango usebenzisa idosi enye. Kuyimfuneko ukwandisa isixa kweziyobisi xa kuthe ukwenza izinto ezintsha okanye amaqela episodic edakumbisayo, kwakunye ukongeza unyango zokuphazamiseka isimo.
Ithamo ngemihla medicament ukuphelisa iingxaki seSkitsofreniya, iziqephu manic nokuphazamiseka kwengqondo isilumkiso uphinda usebenzisa ukusuka 0,005 ukuya 0,020 g, ixabiso leyo ixhomekeke parameters kwezonyango isigulane.
Abadala osezantsi umthamo kokuqala ukuya ku 0.005 g akukhuthazwa, Noko ke, izenzo ezinjalo ziza kusetyenziswa kwizigulana ukusuka kwiminyaka engama-65 ubudala, ukuba kukho ubungozi.
Inkcazelo "Olanzapine Canon" iziyobisi
Le ntshukumo medicament neuroleptic antipsychotic ifumaneka azipilisi isale esingxotyeni salo. Imilo amacwecwe elingqukuviweyo kunye nomphezulu ezimbini khaxa tyheli, imixholo angaphakathi umbala omnye.
Ikhona iidosi ezimbini: kwi 0,005 g kunye 0,01 g olanzapine. Izithako abancedisayo ziquka neselulosi hydroxypropyl kunye endaweni ephantsi, calcium hydrogen phosphate, isodiyam croscarmellose, mannitol, wemagniziyam stearate.
Esingxotyeni yellow Opadry ifilim kwakheka udidi lwesibini, Polyvinyl utywala, macrogol, talc, titanium dioxide, intsimbi oxide.
unyango Drug esimiselweyo Abangaboniyo, ngokubamba nokusebenzisa antirelapse elide izigulane abadala abaneengxaki seSkitsofreniya.
Le unyango lwenziwa monotherapy kunye ulungelelwaniso zidityaniswe kunye compound lithium kunye luhlobo ngamandla izigigaba manic okanye exube bipolar disorder, ezo amabinzana kunye ngezigaba natshintsha ngokukhawuleza ngengqondo kunye. Amayeza ukuthintela kophindo kubantu ukuphazamiseka ngokweemvakalelo, ukuba ichiza kwanceda ukumelana nqanaba mania.
Xa unyango abadala nokudakumba okubangelwa ukuphazamiseka ngokweemvakalelo, kwakunye eliyeza degree edakumbisayo isitali "Canon Olanzapine", indawo neuroleptic, inokudityaniswa arhente equlethe fluoxetine.
It ithathwa ngomlomo, lithe kwizidlo. Guide icebisa ukuba idosi kwezonyango le medicament, nto leyo namhla, inani 0,005-0,020 uthetha akhethelwe ngamnye ukuze isigulane ngasinye kuxhomekeka iimpawu zonyango.
izifo seSkitsofreniya omdala aphathe initial amayeza ongaka mihla 0.010 g lulungiselelwayo kwangoko.
Imeko bipolar disorder mania etsolo ukuphelisa idosi yemihla ngemihla ichiza ukuya 0,015 g okanye 0,010 g olanzapine kudityaniswe arhente equlathe ion lithium okanye valproic acid.
Ukwenza ukusetyenziswa kwengqondo ngexesha Umthamo sokuqala ngemihla oluqhutywa izigulane 0.010 wenziwa ukuba yokwamkela medicament ngenxa mania etsolo, kufuneka uqhubeke ukusebenzisa imithombo mali efanayo.
izifo depressive ezinxulumene izigulane abadala bipolar disorder iphathwa kunye indibanisela 0,005 g kunye 0,020 g ngamalungiselelo olanzapine fluoksetinovyh elawulwa ngokuhlwa.
ukusebenza Antidepressive beziyobisi wabonakaliswa isixa ukusuka grams 0,006 ukuya 0,012 kunye nomthamo avareji yonke imihla ngo-0,0074 g amachiza fluoksetinovyh isusela ukusuka 0,025 ukuya 0,030 g Ukuba kukho imfuneko, kunokwenzeka ukuba kuhlaziywe wemithi omabini amachiza.
uhlobo therapeutic izinzile ndidandatheka isuswe indibanisela 0,005 g kunye 0,02 g iindlela olanzapine fluoksetinovyh lulungiselelwayo kanye ngokuhlwa.
Inkcazelo "Zyprexa" iziyobisi
Le neuroleptic eveliswa azipilisi isale esingxotyeni salo. Kukho ekuqulunqeni idosi ezine: 0,0025 kwi 0,005, 0,010 kwaye 0,0075 ngenxa x, y ezo notation efanelekileyo phezu «Lilly 4112», «Lilly 4115», «Lilly 4116», «Lilly 4117".
izithako baphola ngohlobo lactose, hydroxypropylcellulose, crospovidone, microcrystalline uhlobo neselulosi nesakhiwo abunjwe ngayo amayeza wemagniziyam stearate.
Amacwecwe zipakishwe ngendlela namadyungudyungu zizele 7 pack iqulethe 4 contour ukuphakheja.
Kukho kwakhona ifom owayevunyelwe-ezomisiweyo, yenzelwe eyimveliso kwezisombululo intramuscular. Yellow ulwelo oyidlayo 0.01g wangumqulu oyincwadi ejolise ngqo yentsha. components Engasebenziyo zithathwa monohydrate lactose kunye tartaric acid.
Ichiza liveza ukusebenza antipsychotic.
Eyona nto elikhutheleyo medicament uziphethe ngathi ligand elibophayo kunye serotonin, dopamine, m-choline, H1-histamine kunye alpha1-receptor izinto ezakhiwe adrenozavisimymi. Olanzapine kunempembelelo uyakhetha ngobume ingqondo.
Drug "Zyprexa" umyalelo kwi isicelo ucebisa ukusebenzisa ne zigaba enamandla ukuphazamiseka seSkitsofreniya kwaye ngengqondo ukuba zihamba ngemiqondiso ecacileyo iimfeketho zokufeketha, nemibono, ukuphazamiseka ingcinga, elwayo, isimo sengqondo ezingaqondakaliyo okanye udidi elibi ngohlobo ngaphandle ngokweemvakalelo kunye nezentlalo, ukuphazamiseka ye-apparatus kwezwi. Iyeza iboniswe ukususa iimpawu zasesekondari Uthando okubangelwa ukuphazamiseka seSkitsofreniya.
Icwecwe "Zyprexa" yemiyalezo icebisa ukuba ukusela ngomlomo, nangaliphi na ixesha. Unyango lwangethuba idosi enye ngu 0,010 g Emva idosi yemihla ngemihla isusela ukusuka 0,005 ukuya 0,020 g, apho ebotshelelwe picture nomqondiso.
Intramuscularly zenyuse amayeza, ukuba kukho imfuno engxamisekileyo ukumisa i excitation lengqondo umlinganiswa abantu schizophrenia, ukuphazamiseka kwengqondo Uthando kunye ne-dementia.
Phambi ukusetyenziswa, lo lyophilisate leyo exutywe 2.1 ml injectable zolwelo medium. A isisombululo esicacileyo unomona ebengezelayo.
Le uchulumanco ukoyika disorder seSkitsofreniya kunye disorder awasuse nganye-umthamo 0,010
Xa sicinga ngoku isigulana enyangayo, ulawulo ngokuphindaphindiweyo idosi 0,010 g eyenziwa emva min 120 ukusuka isicelo yokuqala kunye 0,010 g ilandelayo ziphele emva kwemizuzu 240 ukusuka yesibini isicelo.
Ukuba ufuna olusa phambili iziyobisi "Zyprexa" yisa unyango uhlobo yayo tablet kunye umthamo ukususela 0,005 ukuya 0,020 g
Ukuyaluzela sengqondo esixhalabisayo isuswe nedosi enye intramuscular ka 0,0025 Ngokuqwalasela umfanekiso bezonyango kwisigulana, ulawulo idosi 0.005g lwesibini olwenziwa emva kwemizuzu 120 ukusuka isicelo yokuqala.
lencazelo "West Zyprexa"
Kukho medicament "olanzapine" analogs ukuba ziveliswa ngokohlobo lomgubo ngu 0,405 g olanzapine xa ezineengqayi ngesirinji zesinyibilikisi inaliti.
Lithetha "Afrika United Zyprexa" libhekisela antipsychotic msebenzi amachiza neuroleptic.
Amayeza ofihla ukonakala, isetyenziselwa ukugcinwa kunye ixesha elide unyango lwe protivopovtornogo seSkitsofreniya kunye notshintsho sengqondo iimpawu ze-high isivuno ngohlobo iimfeketho zokufeketha, imibono hallucinatory kunye flattening ezimbi iimvakalelo, sisazama indlela izixhobo kwimiphimbo.
Amayeza ngayo iziqephu kakhulu manic kwaye ezidibeneyo ukuphazamiseka ngokweemvakalelo, ngexesha apho iimpawu kunokwenzeka ngengqondo kunye utshintsho ngokukhawuleza ngokwamanqanaba.
oyidlayo Initial ngemihla isetyenziswa yi 0.010 okanye 0.015, ukuba yonke imihla mabaphakelwe ichiza esikhethiweyo ukuba isigulane ngamnye, kuthathelwa ingqalelo umfanekiso lwezonyango. Ezisetyenziswa umthamo enyangayo yemihla ngemihla ukususela 0,005 ukuya 0,020 g
Ukwandisa idosi ichanekile kunokwenzeka kuphela iziphumo ngophengululo. Ukwandisa imali ichiza luqhutywa ngokwamabakala, yonke imihla.
izigulane abadala, idosi sokuqala yonke imihla phambi umsebenzi sezintso elanele wesibindi amisele 0.005 g
analogue iindleko
asolwa elikhulu antipsychotics ukuvumela ukuba ukhethe ichiza ekunene, leyo ofanelekileyo umgangatho kunye neendleko. Imithi "Olanzapine" ixabiso elincinane kakhulu. Packaging iipilisi zingathengwa ngenxa engange-290.
ixabiso "Zalasta" Drug sivela 1370 engange.
indlela ibiza ingqalelo ipilisi "Zidis Zyprexa." Kuba iphakheji imveliso kufuneka ahlawule 2370 engange. Ixabiso analog of "Ku-Tab Zalasta" ngu 1075 engange.
On amayeza "Zyprexa" ixabiso yadla ezimbi. A pack iipilisi 28 ixabisa 4760 engange.
Ngokwamaqela ahlelelekileyo ziya kufumaneka iziyobisi "Olanzapine", nto leyo iqhezu ixabiso.
Views ezigulane
Malunga amayeza "Olanzapine" ncomo unokuviwa kuzo ebezintle nezo zingentle. Abaninzi isiyobisi kuyanceda ukumelana kokudakumba kunye nokunciphisa inani iingcinga ezimbi emva kweentsuku ezimbalwa unyango. He kubhekwa enye amandla neuroleptics, leyo luthoba isigulane, umatshini uloyiko namaxhala.
Phakathi bobubi ayikhuphi iziphumo ezingafunekiyo enxulumene kunye linyuke emzimbeni, oko kukhokelele ekwandeni ubunzima emzimbeni isigulane. Somnolence, asthenia syndrome, isiyezi, igazi intolerance lingehla uxinzelelo uhlobo ukuphuhlisa inyama ithambile ukudumba kwaye kome ngenwebu yangaphakathi.
Ngokuba ezinye izigulane, nkqu igcuntswana leyeza iyeza i sine eyomeleleyo, ukusuka apho balala iiyure ezili-12 ngosuku.
Umzimba womntu ezahlukeneyo, kunjalo, yaye amacwecwe ngendlela eyahlukileyo ukuze isigulane ngasinye. Zokukhetha izixhobo ezifanelekileyo kufuneka udibane nogqirha.
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