Zempilo, Amalungiselelo
"Brilint": inkcazelo ichiza, lo myalelo. Analog "Brilinta"
"Brilint" - ichiza elo lisetyenziswa kutyando kunye nezifo zentliziyo, njengokuba enzile ankoagulyantnym kunye neziphumo antiplatelet. Kwiimeko ezininzi, isetyenziselwa injongo isiqabu zokuhlaselwa of angina (unstable ifom) kunye neentlungu kobuchopho, kwakunye arhente umbala nxamnye ukopha ngokukhawuleza phambi uqhaqho.
Isakhiwo kunye Nokuhlanganiselwa
Ezikhoyo "Brilinta" 90 mg (kwakhona analog) amacwecwe. aba bahamba kuba neqweqwe ifilim a nombala elityheli. NeMilo biconvex ngeenxa zonke.
Eyona nto iphambili ebonakalayo ichiza ticagrelor. Phakathi okunye umsindo:
- mannitol;
- wemagniziyam stearate;
- calcium hydrogenphosphate;
- sodium carboxymethyl starch;
- giproloza.
Lo mboniso, nayo, iquka hypromellose, talc, titanium dioxide, macrogol, idayi (oxide etyheli).
Eyona Ifuthe ichiza
"Brilint" liye amanyathelo antiplatelet, ngamanye kuthintela udibaniso lwe egazi. Ngenxa yokuba eli candelo iziyobisi engundoqo esebenzayo - ticagrelor - zegazi balahlekelwe ukukwazi ukunamathela kunye, yaye ngaloo ndlela zenze amahlwili.
Uhlolisiso ukuqinisekisa into yokuba indlela "Brilinta" ngempumelelo ngakumbi xa zidityaniswe ne salicylic acid. Analogichinye imvume kunye malunga analogu "Brilinta" - "Plavix". Kwezi mvavanyo ababandakanyekayo izigulane kunye nesifo sentliziyo kumaqela yobudala ahlukeneyo, kwaye uthathe ingqalelo yokuba ubunzima lwabo, isini.
Eyona njongo iphambili unyango usebenzisa imveliso uthe - ekunciphiseni ubungozi yokufa, ezinokuthi ingabangelwa ukungasebenzi le nkqubo sentliziyo, ingakumbi sifuba angina kunye iposi engabalulekanga.
Ubungqina obubonakalayo buxela
Reception "Brilinta" kuboniswa kwimeko imfuneko ukunciphisa igazi ekunqandeni, kuquka ukuthintelwa iingxaki sisifo sentliziyo ngohlobo thrombosis kunye thromboembolism. Kungenxa yoko le nto kusifikeleyo oku ichiza eboniswe:
- angina ezingazinzanga (Le ngezifo luphawulwa ukonakala igazi ukusasazwa ukuya izihlunu intliziyo, nto leyo enokusongela engabalulekanga);
- iposi engabalulekanga (ukufa inxalenye intliziyo);
- ukwenza imisebenzi zotyando ezityeni coronary kwemisipha intliziyo (ngexesha ungenelelo percutaneous coronary, okanye Uqhaqho kwimithambo esa igazi).
Ukongezelela ubungqina ngqo, ukuba "Brilint" ngokubona igqirha abanokutyunjwa ukuze sinciphise thrombosis kwezinye iimeko lwezidumbu, njengaxa dissemirovannom coagulation intravascular.
Izimo
Kukho inani iintsilelo, apho ukusetyenziswa "Brilinta" akuvumelekanga. Ezi ziquka:
- isici, kuquka hypersensitivity ukuya into esebenzayo okanye koponentu ubuncinane enye eyongezelelweyo;
- ukopha esebenzayo, ethwele zophendlo lwezifo;
- imilo stroke haemorrhagic ukuba wachukumiseka ngaphambili;
- ukunciphisa umsebenzi hepatocyte, apho iphuhlise sisibindi;
- ulawulo iziyobisi, inyathelo engundoqo iyileyo sikuko inhibition ye enzyme CYP3A4 ( «clotrimazole," "Ritonavir", "nefazodone");
- Abantwana ukuya ku 18 ubudala;
- ngethuba lokukhulelwa zisanyisa.
Xa engekho Izimo kufuneka ukuba phambi kokuba uqale unyango kunye eli chiza.
Imiyalelo yokusebenzisa
Thatha "Brilint" kufuneka ibe ngaphakathi lonke, iyeza kufuneka ukuhlafunwa. Ukusetyenziswa ichiza izimele ngexesha ekudleni. Tablets ndingasela imali encinci bolwelo.
oyidlayo okunikezelwe: 1 ipilisi nganye ngemini. Kubalulekile ukuthatha iyeza yonke imihla ngexesha elifanayo.
Ikhosi unyango kunye nokusetyenziswa 'Brilinta "(ibambela zingenziwa elide) kufuneka uqale idosi kabini (amacwecwe amabini ngosuku lokuqala), uze uye nedosi enye ye-90 mg. Kwimeko ukwamkelwa ichiza kufuneka asebenzise umthamo kabini. Ngosuku olulandelayo emva kokuba baqale ephosiweyo lolwamkelo oluqhelekileyo "Brilinta." Noko ke, iimeko ezinjalo kufuneka kuphetshwe.
I-avareji ubude unyango - iinyanga ezili-12.
Ukongeza, i acetylsalicylic acid ngaxeshanye kucetyiswa.
imiphumela emibi
Phakathi ezibonisa Nedlac abafumana ihloniphekile:
- Ukuncitshiswa ngamandla kakhulu legazi amahlwili kunye nophuhliso wopha ngokungaqhelekanga;
- ziyabagulisa;
- isicaphucaphu;
- ukubuyisa.
Xa iziphumo ebezingalindelekanga ichiza kufuneka imiswe ngoko nangoko.
libanda
Kwimeko ezi mpawu zilandelayo zingenzeka abafumana amathamo eyandisiweyo ichiza:
- isicaphucaphu;
- ukuqumba;
- ukopha;
- ukuphazamiseka intliziyo.
Xa kwenzeka kufuneka uyeke ezithatha ichiza, ukuba lavage esiswini amathumbu, kunye nonyango nomqondiso.
analogs
Xa nakwenzeka ezithatha ichiza kufuneka ukwazi oko ukubuyisela "Brilintu". Phakathi nabalingani ezingundoqo out:
- "Zilt". Eli xabiso "Brilinta" Togu yahlukile, kodwa ifuthe omabini amachiza ezifanayo kwaye ejoliswe ekuthinteleni thrombosis. izithako ezisebenzayo i clopidogrel. Le zibonisa ukuba ukusetyenziswa mali iposi engabalulekanga, coronary syndrome, stroke, fibrillation atrial, coronary okklyuizonnaya kwemithambo. "Zilt" iphawulwa nempembelelo kwicala esinqabileyo.
- "Plavix". "Brilinta" okanye "Plavix" - kokona kulungileyo? Xela ukuba nakanjani na. La machiza into esebenzayo ezahlukeneyo, kodwa isiphumo ezinaso efanayo. Oku kuvumela ukuyeka ikhondo uthomalaliso enye indlela ukuqhubeka unyango kunye nenye. Togu "Brilinta" "Plavix" wabelwe ukuba izigulane abo nesenzeko atherosclerotic ezichongiweyo, izigulane emva isifo sentliziyo kunye stroke. Le ichiza analog nayo zitshiphu. Yintoni ukukhetha: "Brilinta" okanye "Plavix". Kukuphi na okulunge ngakumbi? Xelela ugqirha.
- "Lopirel". Le Togu "Brilinta" enziwe kwi kwisiseko clopidogrel, nto leyo esisizathu sokuba isenzo sibhekiswe zegazi, ukuthintela ukuba lihlale ndawonye. Ngokungafaniyo nezinye iindlela, "Lopirel" kungachaphazela ukusebenza kwe-luvo, izifo, inkqubo musculoskeletal, kwakunye hematopoiesis. Ngaphezu koko, kubalulekile ukukhumbula ukuba eli amachiza analogu "Brilinta" ayikho yokuqala, kwaye generic, oko kukuthi ikopi "Plavix".
Ukongeza kwezi analogue kuvunyelwa ukusetyenziswa nezinye iziyobisi kuba nemiphumo efanayo, kodwa zahluke indlela yokusebenza ( "Cardiomagnyl", "Aspekard", "aspirin-Cardio").
Imigaqo nemiqathango yokugcina
Impilo "Brilinta" (izimvo ngayo phantse yonke HIV) engama-2. Ngoko kuyimfuneko ukuba bagcine ulawulo lobushushu (igumbi apho arhente egcinwe kufuneka ibe izidanga ngaphantsi kwe-30, apho kufuneka kungabikho kukhanya kunye ukufuma). Ukongeza, i-sixhobo kufuneka ukhuselwe ebantwaneni.
Khumbula ukuba zonke izithuba zengqesho kufuneka baziphathe ugqirha.
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