Zempilo, Amalungiselelo
Ichiza "Triftazin": imiyalelo ukusetyenziswa, ixabiso, analogs, ncomo. Libanda, imiphumela emibi, kunye nokupheliswa "triftazin"
"Triftazin" umyalelo Drug eya kuthi ichazwe ngokwenkcukacha kweli nqaku, igqalwa enye amayeza kakhulu antipsychotic. Ukusetyenziswa kweli chiza lu dityanisiwe ubuqili ezininzi ngokwemiqathango idosi ixesha unyango.
Inkcazelo yokulungiselela, ukwakhiwa
Ngokutsho ichiza iqela kuyiphi "Triftazin" libhekisela isiyobisi antipsychotic kunye nempembelelo ngokukhawuleza anti-emetic olomeleleyo. Eyona nto iphambili esebenzayo yikhompawundi evela kwiqela phenothiazines - trifluoperazine, leyo asichaphazeli nje kuphela kwinkqubo luvo, kodwa awo peripheral, ngaloo ndlela, enyanisweni, ngandlela antiemetic.
A Isisombululo ukuba isitofu yi ulwelo ecacileyo, enemibala, akukho ivumba bokuhlala kunye nemvakalo. Tablets "Triftazin" elirhangqiweyo, kugalelwe oluhlaza, ekuqa- emhlophe okanye phantse emhlophe.
Release ifomu, imiqathango kunye neemeko yokugcina
Medicine "Triftazin" impendulo kumagqirha malunga apho phantse sisoloko eyakhayo, kufumaneka ngeendlela ezimbini idosi: njengesisombululo ngenxa inaliti kunye neepilisi. Umxholo wenkqu esebenzayo ampule nganye kunye nesisombululo 0.2% (2 mg 1 ml isisombululo). Le ampoules zipakishwe ngendlela iibhokisi kwi iziqwenga-5, 10, okanye 100 kunye ngemela ampoule ezizodwa kunye nemiyalelo yokusebenzisa iziyobisi.
Emacwecweni "Triftazin" ubuncwane esebenzayo uqulathwe isixa 0,005% (0.5 mg). Bona zipakishwe namadyungudyungu zizele-10, nto leyo, zingafakwa kwiibhokisi zekhadibhodi nezijungqe 4, 5 okanye 10 nganye. Kwakhona ifomu oyidlayo ekhoyo kwizikhongozelo zeglasi emnyama okanye iplastiki emhlophe ngaphaya kwawo, equlethe amacwecwe-50 okanye 100.
Impilo zonke iifom idosi ichanekile iminyaka emi-3. Ukugcina amacwecwe kunye nemiyalelo "Triftazin" solution zokusetyenziswa ekucetyiswa kwindawo epholileyo kunye umoya olungileyo. Awukwazi ukuvumela ukuba iipakethe amayeza ukwalathisa ilanga okanye ulwelo. ayikhuthazwa ukuba ichiza emva komhla wokuphelelwa.
iipropati amayeza "Triftazin" iziyobisi
Makhe siqwalasele iimpawu ezingundoqo ichiza "Triftazin". Imiyalelo yokusebenzisa (lwaseburhulumenteni) inika ulwazi olunzulu malunga indlela yintshukumo engekho mthethweni esebenzayo kwi zemizwa ingqondo kwaye i luvo vagus kwi gastro-emathunjini phecana. Ngokomzekelo, ithi trifluoperazine PMD iibhloko zemizwa ingqondo kunye receptors D2 kwi kwiCerebellum. Ngaphandle kweli neuroleptic nako ukubonelela i Alpha-adrenoceptor ivalela ukusebenza, oko kukuthi, nempembelelo esisebenzayo uxinzelelo lwegazi, ezehlisa kuyo.
Trifluoperazin wafunda kakhulu ngokwaneleyo ngokwemiqathango pharmacokinetics, kunjalo, wazi kakuhle ukuba ngenkuthalo ubotshiwe kwiiproteni plasma (ubuncinane 80%). mechanism coupling ukubola ukuba metabolites njengoko ufundwa kancinane. Kukhuthaza ichiza ukusuka ephilayo kwenzeka ubukhulu becala nge nezintso, inxalenye encinane into esebenzayo kunye metabolites zayo imveliso ngokusebenzisa emathunjini (in inyongo).
Ubungqina obubonakalayo buxela
Ekubeni le ncwadana intshukumo "Triftazin" ukulungiselela uqeqesho ngokucalula nokwahlula njengoko antipsychotic, uluhlu lwezifo apho kufanelekile ukusebenzisa, iquka iintlobo ukuphazamiseka kwengqondo. Phakathi kwabo - schizophrenia, ukuphazamiseka lengqondo, ixhala kunye ukucalulwa (uloyiko ongalawulekiyo esilawulayo). Ngaphandle ichiza isetyenziselwa ukunyanga emesis asibangwa izifo zesisu.
ekhuselekileyo indlela ucinga indlela yaye ingaba zonke iindidi izigulane zingasetyenziswa "Triftazin"? Imiyalelo yokusebenzisa, iingcali yokwenene kunokwenziwa isigqibo sokuba kuyimfuneko ukuba ichiza kuphela emva kokuba kwaqhutywa uphando olubanzi, njengoko kukho inani imiphumela enobungozi kunye Izimo. Ngaphandle kokuba akhululwe ichiza ngaphandle kagqirha, ukuba isigqibo kokungeniswa ayikho imfuneko.
Izimo
Ngelo amacwecwe kunye nesisombululo for "Triftazin" ukuncuntswa Izimo kusetyenziso ukuthini nakwenzeka lokusetyenziswa kwazo. Phakathi kubo bazithumele kudakumbo inkqubo luvo okanye ukuba khokhoma. Ukongeza, ichiza "imiyalelo Triftazin 'ukuba ukusetyenziswa ayikhuthazwa ungenisa izifo zentliziyo, isibindi nezintso, inkqubo hematopoietic. Inqanaba kwesifo kunye ubukhulu ke lawo ukudlala indima ebalulekileyo. Into yokuba kukho inani imiphumo ukwamkelwa iipilisi kunye nesisombululo "Triftazin". ziziphumo ebezingalindelekanga, nto leyo eza kuxoxwa kamva, ngokwabo zinzima kakhulu, kwaye ubukho comorbidities ukuze bandiqumbise nemiphumo nokuba nzima ngakumbi umguli.
Kukwacetyiswa kwakhona ukuba ukusebenzisa isixhobo linembali kukwalisa wengxenye iziyobisi.
Ukusebenzisa i "Triftazin" ngexesha lokukhulelwa
Amayeza esebenzayo kweziyobisi "Triftazin" (reviews of oogqirha ziqulathe ngayo ulwazi oluninzi ngokuxhasa) kunefuthe elibi ekukhuleni kosana olungekazalwa. Ngoko ke ngoko kucetyiswa ukuba ukuthatha amachiza ngexesha lokukhulelwa. Isibakala sokuba trifluoperazine into esebenzayo labonwa kwizihlunu foetal kwiindawo ezixinene kakhulu amathamo zonyango. Ukuba kuphakamisa isethi ezibuthathaka ubunzima ezingekazalwa, nokwandisa amathuba iziphene ezahlukeneyo ekukhuleni kwakhe.
Drug "Triftazin" (analogs ukwimo esebenzayo kubalulekile ukuba uthathe ingqalelo) ayikhuthazwa kwaye phindeke amabhinqa izithako iziyobisi ezifumaneka ngobisi lwebele. Nokuba umama akayi onokuwubukela naziphi na iziphumo ebezingalindelekanga, usana kwixesha elizayo sisenokujamelana neengxaki ezifana tardive zeDyskinesia kunye nokudideka.
imiphumela emibi
Njengoko kuchaziwe ngaphambili, ichiza "Triftazin" kunokubangela eziliqela reactions ezibi inxalenye phantse onke amalungu kunye neenkqubo. Ubukhulu becala into esebenzayo ichaphazela luvo yomguli, nto leyo ethetha ukuba isabelo yengonyama yeziphumo ebezingalindelekanga lwenzeka kulo. Okokuqala, ziquka izenzakalo ezifana iingcangcazela, aqaqambayo entanyeni kunye nolwimi, kutheni ukuze slurred (reactions extrapyramidal). iimpawu zeDyskinesia tardive kuvela rhoqo, sokulibala, akathisia, kunye nezigulo yawo.
Ukusabela zixhaphakileyo evela luvo central zibangelwa ukuthathwa "Triftazin" iimpendulo ichiza ekuthiwa ukozela, isiyezi kunye nelahleko nokucaca umbono. Ngokuqhelekileyo ezi mpawu zisenzeka Ngosuku lokuqala emva kokuqala unyango ngamachiza.
Yintoni enye kunokubangela isisombululo wanyakenye ngenaliti okanye tablets "Triftazin"? ziziphumo ebezingalindelekanga, ngokutsho ubungqina izigulane kunye amagqirha, ngokufuthi kuchaphazela kwinkqubo yokwetyisa. Oku kubonakala ngohlobo lomlomo owomileyo kunye anorexia. Kwakhona, ngokufuthi kukho iingxaki kunye nokusebenza eqhelekileyo esibindini. Ukongeza, ukubonakala uxabane kunokwenzeka yabangxamayo eluswini, amenorrhea, agranulocytosis.
oyi
Imiphumo ezibi ikhankanywe apha ngentla nga ncitshiswa yi unyango kwangumqondiso okanye uhlengahlengiso idosi. Rhoxisa "triftazin" iyafuneka kuphela xa kukho ukuphazamiseka kakhulu kwiisistim ilungu yesigulane. Ngenxa yoko, nathi ingqalelo ubuchule kunye neendlela zokulahla ezisisiseko okanye ukunciphisa abasabela engafunekiyo ukuba ichiza.
Xa Barr okanye nokuxutha izinto kwiimeko ezininzi, iingcali uthatha isigqibo ukunciphisa ngeedosi ezithathwe sisigulane okanye ekumeni reception kwakhe okwethutyana. Kwiimeko kakhulu angafuna unyango kunye namachiza antiparkinsonian, barbiturates okanye iziyobisi caffeine (ulawulo emthanjeni).
Xa iimpawu abuthethileyo of ukuphuthelwa okanye motor disinhibition, ukuphazamiseka ayikhuthazwa ukunyusa idosi yokuqala. Ngokwesiqhelo kwiintsuku nje ezimbalwa umzimba wayethimb ichiza elitsha, kwaye iimpawu ezibi iyanyamalala kancane. Kungenjalo, oku kufuna unyango ngamachiza "benzodiazepine" okanye "Propanolol".
Loo urhulumente zeDyskinesia tardive, okhankanywe phakathi iziphumo ebezingalindelekanga xa uthatha "Triftazin" iziyobisi, ncomo kuzo ziza kuchazwa koku, ngokufuthi ikhula ngenxa yokusetyenziswa ixesha elide ichiza okanye kamsinya nje emva kokuba ukurhoxiswa kwayo. Iingcali uqaphele ukuba zeDyskinesia (tardive) adla sifo kwizigulana abadala.
Ezinye iziphumo ebezingalindelekanga okubangelwa ukuthathwa a medicament ingahimbiselani iintshukumo ezifana nokulawula izithuthi kunye neendlela ezintsonkothileyo. Ngexesha unyango "triftazin" Kungcono ukuba ayeke kubo.
Izikhokelo iidosi kunye neendlela nokulungiselela Hour
Nesilinganiso ogqitywe oyingcali ngokwesiseko yomguli ngamnye, imeko yakhe phambi izifo ezihamba. ithamo ubuncinane "Triftazin" ichiza esuke ngexesha kwangoko unyango. umyalelo tablets siyalela uthathe 1-5 mg amaxesha 2 ngosuku (izigulane abadala). Kwiiveki ezintathu ezilandelayo, idosi ebegqwese ukwanda nokutshintswa ku 45-60 mg ngosuku. Le mali kufuneka kwakhona kwahlulwa zibe ngamanqanaba amathathu.
Kuba unyango kwabantwana kuqhelekile ukusebenzisa ngeedosi ezincinane ichiza. Ekuqaleni unyango maningabi sathabatha ngaphezulu kwe-3 mg ngosuku (ngokwamanqanaba 3). Ukuba kuyimfuneko, kwaye xa kungekho yeziphumo ebezingalindelekanga ngokukhawuleza kwizigulo pamo lanyuka ukuya 6.5 mg ngosuku.
Inaliti "Triftazin" imele ukwenziwa intramuscularly ngamathuba iiyure hayi ngaphezulu kwe-6. Le idosi yemihla ngemihla abadala kunye ubuninzi-10 mg. Abantwana ibonisa umthamo 1 mg ngosuku, yahlulwe yaba iinaliti ezimbini, ngamathuba esingekho ngaphantsi kweeyure ezingama-12.
Sinqwenela ukutsalela ingqondo yomfundi ukuze yokuba unyango nalo eli chiza, kungakhathaliseki uhlobo idosi kufuneka kwenziwe phantsi kweliso gqirha. Nguye isigqibo malunga notshintsho idosi i kwizigqibo amayeza "Triftazin". Libanda, xa isetyenziswa kakuhle, lithetha ngathi akunakwenzeka. Ukusetyenziswa olungagunyaziswanga ichiza, okanye utshintsho idosi ekucetyiswa ngendlela enkulu kunokukhokelela imiphumo engalindelekanga.
imithi
Onke amachiza bakholisa ukuba basebenzisane kunye nabanye. Iipilisi kunye "Triftazin" isitofu kulo mba kungekho ngaphandle. Ngokuqhelekileyo, iingcaphephe ukuthathela ingqalelo imiba emininzi ezichaphazela ukusebenza ngayo ukusetyenziswa kweli chiza. Ngenxa yoko, imithi eziqulathe ethanol (isiraphu, tinctures kunye ezifana), CNS depressants ukuze yandise iimpawu "triftazin", kwaye kananjalo kuchaphazela iinkqubo nokuphefumla ngokungalunganga.
Kunye neziyobisi ukunciphisa uxinzelelo lwegazi, tablet okanye isisombululo "Triftazin" kufuneka isicelo ngononophelo kakhulu kangangoko kunokwenzeka uphuhliso hypotension ahlekise intolerance.
Asidi kunye nee-arhente antiparkinsonian igalelo kukufakwa elithotyiweyo le iingqalutye into esebenzayo "Triftazin" ukusuka wokugaya kwaye, ngenxa yoko, ukunciphisa ifuthe ichiza.
Le nefuthe elibi ayibonileyo-isicelo nokubambisana neziyobisi xa idibene neetyuwa Lithium. Ngokutsho ingcaciso efunyenweyo, ukuhlanganiswa elinjalo igcwele nophuhliso iimpawu extrapyramidal iqapheleka kunye nokwanda neurotoxic ukusebenza trifluoperazine.
Izimvo amayeza "Triftazin"
ezininzi zizama ukufumana reviews ngayo phambi kokuba uqale ezithatha ichiza. Medicine "Triftazin", ukugweba la magqabaza leengcali, igqalwa omnye kakhulu ngempumelelo. Ngelo xesha, ukuba uqaphele ukuba ulwimi ezithatha ichiza unokuba nefuthe elibi hayi kwi ebonakalayo kodwa isimo sengqondo yomntu.
Kuba abo izigulane usibonisileyo nangokwamkela beziyobisi, kwiimeko ezininzi ekuphela kwendlela ukuphila ubomi obuqhelekileyo. Kakade ke, ayikho ngaphandle iziphumo ebezingalindelekanga. Kodwa, njengako manani, zonke iimpawu ezingemnandi shwaka phakathi iiveki ezimbini emva kokuba unyango.
Imibono malunga izigulane 'Triftazin "amayeza igalelwe. Enye ngokwenene wanceda, ngoxa abanye kunzima kangaka ukuba ukulunyamezela side effects kwadingeka bayeke esisixhobo. Amaxesha amaninzi abathengi zibonisa ukubonakala ukudinwa, silale kunye ubuthathaka jikelele. Kwiimeko ezinqabe kakhulu, izigulane yawa zibe kwimeko apho abafuni ukwenza nkqu iintshukumo ezininzi ezingundoqo.
Abafazi, ngokungafaniyo abantu, badla ukunyuka ubunzima bomzimba ekhankanywe ngexesha unyango with "Triftazin". Iingcali athi unxulumano ngqo phakathi le unyango ngamachiza kwaye akukho nzuzo weight. Babecinga ukuba oku kubangelwa kukuhla kumsebenzi motor izigulane ngokuchasene nentsukaphi ulondolozo yokudla yangaphambili.
Awasebenzisa malunga nefuthe iziyobisi, kunye noogqirha kunye izigulane ziye wabona ukuba okunene kubelula okanye asuse zonke iimpawu zesi sifo ngxabano.
Analogs neendleko ichiza
Ngoko ke, wabancina imiba ebalulekileyo ngokusetyenziswa "Triftazin" iziyobisi. Apho unayo nokutshintshwa ezilinganayo, okanye ekuthiwa analogs? Kakade ke, la machiza ngeenkalo. Ngoku Antipsychotics ukuvelisa phantse zonke iinkampani zamachiza, kwaye inkoliso amachiza kweli qela zithiwe thaca nelithi "triftazin" (okt kumkhawulela kulwakhiwo). Ezi ziquka "Vespezin" iziyobisi "trifluoperazine hydrochloride", "trifluoperazine hydrochloride", "fluazinam," "Ekvazin", "Stelazin", "Cyclodol" kunye nabanye abaninzi.
Iindleko kula machiza azisoloko efanayo. noogxa bamanye amazwe badla kubiza kakhulu, xa kuthelekiswa ne ichiza "Triftazin", endiwazuze umlinganiselo engange 50-70 pack ngamnye (tablets 50). Ukuba sicinga ukuba ukusetyenziswa kwale sixhobo, ubude unyango, kufuneka ingqalelo ixabiso layo njengomnye okulungileyo ngaphezu analogs amazwe.
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