Zempilo, Amalungiselelo
"Tizin Alerdzhi": ncomo. Kuncipha kwi impumlo "Tizin Alerdzhi": ixabiso guide
Yintoni izigulane malunga ichiza "Tizin Alerdzhi"? Izimvo medicament kuthiwa thaca ekupheleni kweli nqaku. Kuwo uya kufunda malunga nendlela apho isixhobo yenziwa, wobeka phi kubiza, yintoni na into iqulethe kukodwa, yaye zintoni na iimpawu.
Ubume, inkcazelo, ifomu kunye nokupakishwa
Ngeempumlo uwisa "Tizin Alerdzhi" zimele ukunqunyanyiswa emhlophe yohlobo olunye. Eyona nto elikhutheleyo medicament yi hydrochloride levocabastine. Ngaphandle kwalo, ichiza ikwaquka izithako ezongezelelekileyo ezifana sodium hydrogen phosphate, propylene ethers, hypromellose, isodiyam monohydrate, polysorbate, benzalkonium chloride, ngamanzi okuhlamba kunye disodium edetate.
Uwisa "Tizin Alerdzhi" imfundiso leyo ifakwe kwi ibhokisi eveliswe nengqayi ye ml-10. Yakhiwa polyethylene, kwaye mayixhotyiswe isitshizi (kuba lula) kunye ikepusi nokhuselo olukhethekileyo.
Pharmacology kuthetha
Ukulungiselela "Tizin Alerdzhi", ixabiso equlethe ngakumbi imele medicament antiallergic. Ngokutsho imiyalelo, amathontsi anjalo nefuthe ngqo kwi uyakhetha blocker H1-receptor (histamine).
Emva kokuba isicelo beziyobisi umguli shwaka phantse zonke iimpawu nokuthimliswa ukuba imvelaphi uyalisa. Kwakhona, eli chiza akubikho ukurhawuzelela kunye nempumlo esihambisayo. Ukongeza, oku kuthintela nangokuthimla uhlaselo.
Bambalwa abantu bazi, kodwa amachaphaza "Tizin Alerdzhi" zingasetyenziswa kuphela ukuba instillation kulo impumlo, kodwa emehlweni. Ngokuqhelekileyo, xa kusenziwa lwamehlo nokuzisebenzisa conjunctivitis komzimba.
Ngokutsho iingcali, isiphumo emva kokuba isicelo medicament kwenzeka emva malunga 5 imizuzu kwaye ithatha iiyure ezili-12.
Pharmacokinetics
Ulawulo Intranasal of medicament (xa isixa-50 g) wendele malunga 30-35 micrograms levocabastine. Ayithandi eliphezulu egazini malunga neeyure ezintathu.
Ukubambana osisiqu esebenzayo kwiiproteni plasma nama-55%. Le metabolite engundoqo (atsilglyukuronid) beziyobisi yenziwe ngexesha glucuronidation.
Isiqingatha lobomi into efana levocabastine, ziiyure 37-40. Oku kwakuthe kwizintso (ubukhulu becala kutshintsha).
ubungqina
Kuba yintoni ukusebenzisa iyeza "Tizin Alerdzhi" injongo? Ukuphonononga baxele ukuba ngamathontsi ezinjalo ngempumelelo azibonakalisa kunye nokuthimliswa uyalisa kunye conjunctivitis. Kwakhona, eli chiza omiselwe hay fever kunye exacerbation rinokonyunktivalnom syndrome.
Izimo
Hlobo luni Izimo kufuneka bazi phambi ngokusebenzisa ichiza "Tizin Alerdzhi"? Izimvo kumagqirha bathi eli chiza aluvumelekanga ukuqesha hypersensitivity wesigulane ukuze sisebenze kunye additive, nto leyo eyinxalenye amathontsi.
Kwakhona, eli chiza ayisetyenziselwa yonyango abantwana abangaphantsi kwiminyaka emi-6 ubudala.
Ngononophelo ngeempumlo kunye neliso amathontsi sele Kucetyiswa ukuba basebenzise abadala kunye nabo abaphethwe ukusilela kwezintso.
Uwisa "Tizin Alerdzhi": imiyalelo yokusebenzisa
kufuneka isetyenziswe njani yokuphatha ichiza? Waye wamiswa intranasally. Abantwana abadala ngaphezu kweminyaka emi-6 kunye nezigulane abadala bacebisa ukusetyenziswa amathamo 2 ichiza (oko kukuthi, 100 micrograms) ethatheni ngalinye kabini yonke imihla.
Ukusetyenziswa kwale nyango kufuneka waqhubeka ukuphelisa zonke iimpawu zesi sifo. Xa wavakalisa neziyobisi iimpawu zesi sifo ingasetyenziswa izihlandlo ezine ngosuku.
Ngaphambi kokuba usebenzise amayeza isigulane livuselelwe ukusula amarhanana evela ukukhetha ezikhoyo uze uphefumle (ngokusebenzisa impumlo) ngethuba lokusebenza kwenkqubo imithi.
umthamo
Indlela kungcwaba ichiza "Tizin Alerdzhi"? Ukuphonononga bathi phambi ukusetyenziswa yokuqala ngezixhobo eziyimfuneko ukuze ususe le chap zokuzikhusela, yaye emva koko izihlandlo eziliqela ukuba cofa umlomo. Ngenxa ukutshiza enjalo umoya kufuneka ibe kutsala "nenkungu". Okulandelayo, faka esatsiba kulo sicatshulwa ngeempumlo nokuzalisekisa namaphephandaba. Ngelo xesha ke kufuneka ukuba aphefumle impumlo yakho.
Phambi kokuba isicelo elandelayo tsakisi kakuhle Shake.
imiphumela emibi
Ngelishwa, kaninzi ingqalelo ichiza ibanga iziphumo ebezingalindelekanga. Ezi ziquka oku kulandelayo:
- isicaphucaphu, ukozela;
- womile, ubuhlungu kuyo inaliti, uvutha;
- intlungu kwingqula nasemqaleni, ukukhohlela, epistaxis;
- udumba isifo ngeempumlo, bronchospasm;
- tachycardia, negazi;
- intloko ebuhlungu, isiyezi;
- ukudinwa, ezidlulayo usi lendawo;
- umkhuhlane.
libanda, iziyobisi
Iingxelo ze libanda, le mali ziye zafunyanwa. Kodwa ke, iingcali zikholelwa ukuba xa ngengozi sihlisa yokwamkela ngaphakathi Isigulana: ukuncipha uxinzelelo lwegazi, omnye umthomalalisi encinane kunye tachycardia.
Ukuze ukuphelisa iimpawu ezinjalo imfuneko abachaphazelekayo ukuba usele izixa ezikhulu zamanzi ukuze kukhawuleziswe zinomgutyulo yi izintso levocabastine.
imithi
Kwizifundo zonyango, impefumlelwano ichiza baligalele kwaqwalaselwa. Kwakhona ezichongiweyo abazange ngcono imiphumela "Diazepam" ngoxa ukusetyenziswa ngeempumlo sihlisa "Tizin Alerdzhi" kwi iidosi eziqhelekileyo.
Indibaniso oku kuthetha nge "erythromycin 'yaye isoenzyme CYP3A4 inhibitors ketoconazole aluchaphazeli entshukumo iparameters levocabastine.
intsebenziswano Local beziyobisi kunye namanye amalungiselelo intranasal wahlolwa, ngaphandle intsebenziswano yawo kunye "oxymetazoline". Ke kaloku, kwanciphisa (transiently) ukufakwa yokugqibela ngeempumlo sihlisa "Tizin Alerdzhi".
izincomo ezithile
Ukulungiselela "Tizin Alerdzhi" (umsebenzisi beziyobisi efunekayo ukuze ukufunda) lungenasiphumo sine kananjalo akusenzi isantya yokusabela.
Ukuba ngaba wehlelwa ukozela isigulane ayikhuthazwa tu into yokuba nenxaxheba kwizinto eziyingozi, kwakunye ukuqhuba iimoto.
Emva kokuphela ichiza akayi ufanele aphoswe kude phandle okanye uhlanganise angcolile. Ichiza kufuneka abekwe kwingxowa kwaye ufake kwi emgqomeni.
Iindleko amayeza kunye analogue
Kangakanani na amathontsi "Tizin Alerdzhi"? Ixabiso eli chiza ayikho phezulu kakhulu. Ungenza kusithenga 210-280 engange.
Ke noogxa, bona kakhulu kunene. Baye izenzo ezifanayo amalungiselelo afana "Vizin Alerdzhi", "Gistimet", "levocabastine," "Reaktin". Noko ke, siyiguqulela iziyobisi "Tizin Alerdzhi" kufuneka ibe kuphela emva kothetha-thethwano kunye nogqirha wakho.
Izimvo kulungiselelwa
Uninzi izigulane ukhe wasebenzisa iziyobisi, eshiya ngaye feedback kuphela HIV. Bathi ingxelo ukuba eli chiza ngokupheleleyo esizibonakalisa xa kuthe iimpawu nokuthimliswa komzimba kunye conjunctivitis komzimba.
Emva kokusebenzisa eli chiza xa izigulane phantse ngoko nangoko yokumpompoza ngeempumlo. Ngaphaya koko, eli chiza kuthintela nangokuthimla.
Njengoko ngokuba bawo, abarhanelwa ziquka ukungakwazi ukusebenzisa amathontsi ngethuba lokukhulelwa ngexesha lokuncancisa. Kwakhona, abantu abaninzi ukhalaze malunga yokuba eli chiza kufuneka ingasetyenziswa xa abantwana ukuya kwiminyaka emithandathu.
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