Zempilo, Amalungiselelo
Analog "Flucostat" (ezitshiphu). Tablets "fluconazole" - ncomo, amaxabiso
Ubuntu ikhona kwi emhlabeni kangangamawaka eminyaka. Ngalo lonke eli xesha kunye nabantu abahlala ngempumelelo azivelele kubekho izinto ezincinane. Abaninzi kubo ayimfuneko ukuze umntu ukuze bajongane neemeko ezahlukeneyo lwangaphandle ndlongondlongo. Kodwa kukho abo inokubangela izifo phantsi kweemeko ezithile. Oko enjalo iquka iintlobo ezahlukeneyo ezincinane ezinzwaneni rhoqo ephethe isoyikiso empilweni yoluntu. Ukuze kujongwane nazo iminyaka emininzi, oosonzululwazi nokuphuhlisa arhente nokubola.
Mhlawumbi kwizikhundla akhokelayo phakathi uluhlu olude izixhobo ezinjalo ichiza "Flucostat". Nangona kunjalo, akukho ziyafikeleleka kwaye ifumaneka ngokude hayi onke amacandelo oluntu. Kakhulu eqhelekileyo nangakumbi iyeza "fluconazole" - nelo ukuba "Flucostat". Zitshiphu (15-30 engange nxamnye 170-300), kunye emininzi ebanzi amanyathelo kweli chiza ayikho ngaphantsi oko, nto leyo analogu.
Yintoni i-fluconazole?
Enyanisweni, i-fluconazole - engundoqo icandelo esebenzayo iziyobisi "Flucostat" - yinto inhibitor esinamandla (into nako isantya okanye ngokupheleleyo ukuyeka naziphi nokomzimba) stem sterols kwiiseli ezinzwaneni. Le into uyakwazi ukumelana ubunzima arhente causative engundoqo mycosis olungenelelayo (zizifo ezingenelelayo unokubangwa amagciwane olungenelelayo, ezo ngokubanzi ezikhuselekileyo umntu inkqubo esempilweni omzimba). Ngaphezu koko, unyango "-fluconazole" olusebenzayo ekubhaqeni Cya fungal, uphawu bendawo ethile (mycosis ikho).
Action emzimbeni womntu
Emva nokudla ichiza ako kakuhle. Ngaxeshanye ekudleni alunasiphumo kwi indlela yalo nkqubo. Emva zokwamkelwa philisi "fluconazole" ngokukhawuleza kwalutyhutyha phantse zonke neencindi zomzimba. Izalathi si zokunikwa eyavela kwi-plasma yegazi, namathe kunye isikhohlela ziyafana omnye komnye. Xa izigulana luhlobo fungal sokudumba kwenwebu yengqondo, amanqanaba fluconazole kulwelo cerebrospinal lifikelela 80% of pokazateya plasma. Amalungiselelo evela emzimbeni womntu kakhulu nezintso. Ekuqhubeni uphando malunga nama-80% ye-dose ezilawulwa ibanjiwe esenjalo kuwo yokuchama.
Ubungqina obubonakalayo buxela
Ukulungiselela "fluconazole" yesikhokelo (ixabiso kuxhomekeke kwiifom ukukhululwa: tablets, njengezingxobo, Ithatyathwe emigutyeni ngenxa zokumiswa yolawulo ngomlomo, isiraphu, izisombululo inaliti emthanjeni) uncoma ukuba uluhlu olubanzi ngokwaneleyo na usulelo ezinzwaneni ezenzeka emzimbeni womntu. Uluhlu kwezifo iquka cryptococcal meningitis (meninges sisifo esibangelwa ngundo), nto leyo inokuba nemiphumela emibi kakhulu ukuba umntu. Kwakhona ezinokubanceda analogu "Flucostat" thrush (candidiasis kusisi), kwaye zonke iintlobo candidiasis lwenkqubo.
Iingcali amisele ichiza kwizigulane kunye nezifo kuyehla njengenyathelo lothintelo. Kwakhona amayeza "fluconazole" wamisela abo usulelo ezinzwaneni emva kokuba unyango ngokwaneleyo ngxwaba umhlaza (unyango radiation, amayeza, cytostatics). unyango zintsholongwane kwakhona kunokubangela iimpawu zezifo ezinzwaneni ekufuneka zilahlwe kuyo nayiphi na imeko.
Ibonisa ukusetyenziswa kweziyobisi emva imisebenzi ilungu esinye. Ikhondo unyango unyango kunye nokusetyenziswa kweziyobisi immunosuppressive nazo kwenza kube yimfuneko ukuba analog olusebenzayo "Flucostat", izimvo zazo ingacaci ngokwaneleyo.
Zonke iintlobo omzimba usulelo ezinzwaneni ulusu (olusisikhokelo pedis kwaye kuquka) kwindawo nasemiphakathweni, onychomycosis (usulelo iinzipho nokungunda), pityriasis versicolor (eziyimibalabala elide okanye esingapheliyo ezinzwaneni of sangaphandle) nazo kwisigaba eziphembelela "fluconazole" iziyobisi. Abantu kabi eqhelekileyo wokugonyeka zinikwa kwimeko mycoses enzulu ngokwasendalweni apha.
Unyango Kucetyiswa ukuba uqale kwangoko, ngaphandle kokulinda ukuba iziphumo zophando kunye nokulima. Noko ke, xa ezi ziphumo ziya kufumaneka, unyango kufuneka ilungiswe. Unyango kufuneka kuqhube okoko nje unyango esipheleleyo ayiqinisekiswanga laboratory kunye nezifundo zonyango kwaye ahlalutye. ukupheliswa ngaphambi kunjalo unyango uya kukhokelela ukwenzeka ezinzwaneni. Kulo mzekelo, kusenokwenzeka ukuba kungafuna ukwandisa amathamo amayeza kunye zobude kwexesha imithi yethutyana, njengokuba uhlobo ezincinane bafumana ukumelana (okukwazi) ukuba kukho into esebenzayo "fluconazole".
Izimo: Ngubani kufuneka ayeke ukuthatha
Medicine "fluconazole" yemiyalezo (ixabiso lincinane noko, kule meko, akukho ngomlinganiselo efficiency) awenzi ukuthatha abantu abahluphekayo ukunyamezelana ngamnye iincindi zalo eziphambili. Musa ukusebenzisa eli chiza ukuze unyango lwezifo ezinzwaneni kwabo abaphethwe ekubonakalisweni komzimba naluphi na uhlobo ku clotrimazole, miconazole, ketoconazole, econazole, terconazole, sulconazole, sertaconazole. ukusetyenziswa azamkeleki ngaxeshanye iziyobisi "fluconazole" yaye "Cisapride" ( "Propulsid").
Ngaba ukuba makwaziswe umvavanyi ngenjongo yokuba bakuthathele ingqalelo kugqirha echaza yokwamkela ingxaki kunye nezintso, nomhlehlo wesibindi, ukuphazamiseka zentliziyo, ubukho imbali ngokwabo okanye syndrome ngayo usapho lwakhe lokuphumla evuthelweyo QT (ukungasebenzi yombane entliziyweni, inokukhokelela ngesiquphe ukulahlekelwa sezingqondweni kwaye ikhokelele ekufeni).
Drug "fluconazole" kunye nokukhulelwa - mali incoko eyahlukileyo. Gynecologists bakholelwa ukuba ukusetyenziswa ithamo elinye single (150 mg) akuyi kubenzakalisa usana. A unyango systemic ngala machiza kunokubangela uphuhliso malformations iziphene emntwaneni.
Ngokutsho uphando, ukusetyenziswa ngeedosi eziphezulu (400-800 mg yonke imihla) ixesha elide ukukhulelwa kwakhokelela ekubeni kukuba abantwana badla ukuphuhlisa ukungaqheleki enqabileyo iziphene: brachycephaly, malformations na igumbi cranial, "inkalakahla", iziphene iziphene intliziyo. Ukuba umfazi akhulelwa ngexesha unyango (Isingxobo okanye icwecwe) "fluconazole", ugqirha kufuneka uqinisekise ukuba kuziswe ingqalelo yayo, ukuba umngcipheko ukuba usana. Ukuba umama elizayo wagqiba ukuba umntwana kufuneka azalwe, ukuba abasebenzi bezempilo kufuneka ngenyameko kakhulu esweni indlela ekhulelwe.
Ngokubanzi, gynecologists bacebisa ukuba abasetyhini abafumana unyango lweNTSHOLONGWANE ezinzwaneni lonke ixesha unyango kukudliwa kukhulelwa olusebenzayo.
Kwakhona, le analogu "Flucostat" - iziyobisi Russian "flucanozole" - musa ukuthatha abantwana abangaphantsi kweminyaka emi-4.
Drug "fluconazole" kunye candidiasis lobufazi
Kusisi candidiasis (thrush) okubangelwa igwele Candida. Le ngundo ekhoyo emzimbeni mfazi uye njalo yaye ngokuqhelekileyo abangela izifo. Noko ke, xa ngenxa yesizathu esithile buthathaka umzimba okanye jikelele emathunjini kunye ikuku kwabasetyhini ukuba anciphise inani iintsholongwane siyingenelo. Apha kwakhona iyasebenza Candida.
Umfutho uphuhliso thrush inokuba eziliqela izizathu. Oku kunokuba yinto eqhelekileyo vitamin ukuswela okanye ukungabikho iihomoni ababhinqileyo sex, ukungatyi ukutya okunesondlo, okanye ntshikilelo rhoqo khulu. mandundu ukuze ube ungenzi nto, enxibe impahla tight okanye impahla eyenziweyo, ukusetyenziswa kweziyobisi zocwangciso hormone okanye iziphumo zonyango kunye antibiotics. Kanti ke, njengokuba oko kusenokubonakala ngathi engaqhelekanga, ichiza "fluconazole" thrush kuya kufuneka ukuba abo bafazi abahlukunyezwayo yi douching okanye izixa ngokugqithisileyo arhente ezahlukeneyo antibacterial esetyenziselwa nokunyamekelwa kwezi esini. Kulo mzekelo, kunye kwamagciwane zixheliwe, yaye zonke izilwanyana luncedo kwinxenye yelungu lobufazi.
Iimpawu zokugula igwele kwamabhinqa imbonakalo obhobhozayo obufana, ukutshisa kunye ukurhawuzelela kwindawo angasese, ukudumba kunye anozizi zangasese, ukuchama kabuhlungu. Phephezela sex ubuhlungu. Nangona kunjalo, ezi mpawu ekhona kwezinye izifo amalungu esini ababhinqileyo. Ngoko ke, ngaphambi kokuba uthathe iziyobisi "fluconazole" ukusuka igwele, kuyimfuneko ukuba ukutyelela ugqirha, iwise uviwo ebanzi kwaye uqinisekise ukuba candidiasis lobufazi, kwaye hayi enye into ofuna irejimeni yonyango ezahlukeneyo kunye namanye amayeza.
Namhlanje, ishishini lamachiza uvelisa iziyobisi kuluhlu enkulu, ezinako ukumelana thrush. Nangona kunjalo, icandelo esebenzayo iphambili abaninzi kubo fluconazole. Le Togu "Flucostat" nakho ukufikelela ngakumbi kuluhlu olubanzi abathengi ngenxa yesizathu esilula sokuba zikhutshwe ngomhla intsimi umakhi zasekhaya Russian.
Ukuthatha le amayeza thrush
Icebo "fluconazole" kuthetha elula ngokwaneleyo. Ukuba sifo sasibonakala okokuqala, yaye lo mfazi ngokukhawuleza ubuyeleyo ugqirha, ukuze ufumane nemiphumo emihle zonyango kunye nokufunyanwa ngokupheleleyo iya kuba yanele nedosi enye ye-drug-150 mg. Ukuze ukulungisa yoko, emva kweentsuku nje ezimbalwa, ungakwazi ukuthatha nkqu tablet elinye okanye capsule. Ipatheni efanayo yamkelwa kunye namayeza "Flucostat". Togu "fluconazole" nje ayibizi, kodwa oko akuthethi kuchaphazela ukusebenza kwayo.
Noko ke, ukuba umfazi uthe uhlobo okondeleyo engenagwele, kwaye ezi izigulane ngoku malunga ne-5%, ngoko isicelo wesekethe "utshintsho Flukonaloza 'kakhulu. candidiasis Chronic kusisi kunzima ukunyanga, kudala waqhubeka, ngokulula mkhuba. Kwiimeko ezinjalo, idosi enye kakhulu enganelanga, kwaye ugqirha wonyula izifundo elide yonyango. Ngokuqhelekileyo, ichiza kuthathwa kabini ngeveki kwiiveki ezingama-2. Ngaphezu koko, zingaphelanga iinyanga ezintandathu kuyimfuneko ukuba ichiza (njengezingxobo okanye tablets) "fluconazole" kanye ngenyanga kwi idosi abangama-150 mg.
Ngokubanzi, ukukhethwa scheme, oluya kubanjelwa kwi yonyango candidiasis kwilungu lobufazi, kuba lilungelo leZiko eliQinisekisa gqirha khona. Ukuba ugqirha kufuneka ukuvavanya ubuzaza imeko yomfazi, ubude impawu yokuqala, ubukho iingxaki zempilo ezinxulumene (badla thrush - yenye zosulelo, izifo ezidluliselwa ngeentlobano zesini kuphela). Emva kokuhlalutya zonke ezi zinto kunye nempembelelo yazo kwendalo umzimba yomfazi, ugqirha uya kukwazi ukukhetha irejimeni yonyango kakhulu ngempumelelo besebenzisa le analogu ethile "Flucostat" ukusuka Igwele (ixabiso kule meko ayibalulekanga).
ziphumo bezingalindelekanga kunokwenzeka
Ngokubanzi, iziyobisi "fluconazole 'Wanyamezela kakuhle nasiphi na isicelo (zombini efakwa kunye ngomlomo). Ngamanye amaxesha ungabona utshintsho ekusebenzeni wesibindi, nezintso, kodwa amaxesha amaninzi oku kubangelwa beziyobisi izigulane kunye nezifo kakhulu ingxaki, ezifana nogawulayo kunye nomhlaza.
Abasetyhini abafumana nedosi enye ye-150 mg ukuba unyango lwezifo obuni, kwaye ngamanye amaxesha sibonakala iziphumo ebezingalindelekanga ezifana iintlungu esiswini, ubucaphucaphu okanye yintloko. Ngobunzulu ngokwesiqhelo wavakalisa ngobulali okanye ukumodareyitha.
Ukususela luvo kwaye ngamanye amaxesha izinto ezifana sokuwa, isiyezi, ukulala lembandezelo, lafa. iphecana zesisu zinako ukuphendula isicaphucaphu amayeza, urhudo, ukugabha, incasa okungaqhelekanga, ukungabi namdla. impendulo kwesibindi ukuba ichiza nalo kakhulu edidayo. Ukuba isigulana Akukho zifo ingxaki kakhulu, ixesha lolwamkelo kunokubangela ukuphazamiseka ngomsebenzi wayo, nto leyo ayavalwa ukususa ichiza. Xa isigulane izifo zinzima kwaye enzima ezinkulu (Lusenziwa leyo baphathwa ngamayeza ezahlukeneyo), eli Togu "fljukostat" (ngaphantsi nokubola ebiza okanye ngaphezulu, ayibalulekanga into, ngokuba icandelo engundoqo esebenzayo - fluconazole) maxa wambi kubangela iingxaki ezinjalo kunye isibindi ezifana hepatitis, cholestasis okanye ukusilela hepatic leyo kwezinye iimeko zingabangela ukufa. Noko ke, umntu athi kakuhle ukuba neziphumo ngcwaba ezibangelwa ichiza anti-ezinzwaneni kukuba imeko engundoqo ithathwa amayeza ezintsonkothileyo.
Iingcali, dermatologists bathi ichiza "fluconazole" kwiimeko ezinqabileyo kunokubangela nerhashalala kuvela ulusu neenwele ilahleko (idla ngokuba ngabo abathabatha ichiza ngaphezulu kweenyanga ezimbini). Emva ukupheliswa la ezingemnandi shwaka.
ngeedosi kakhulu: Implications
Ngaphandle ukusetyenziswa amathamo eziphakamileyo ichiza gqirha "fluconazole" (ixabiso; ncomo kulo mzekelo ingaba sibagxeke) kungakhokelela libanda. Ezi mpawu zixhaphakileyo lidiza of overdosing esinzulu, ngokuqhelekileyo yokuphazamiseka iphecana zesisu (isicaphucaphu, ukugabha, urhudo). unditsho kunokwenzeka kwiimeko ezinzima. Ukuba ukuthathwa zonke ezi mpawu, ichiza kufuneka kurhoxiswa. Ukuba, emva kokuba lo uzibonakalisa i libanda, akukho wayeka, kuyimfuneko ukuba udibane nogqirha.
Unyango kulo mzekelo zangathi ziziikopi zezo ukunciphisa kukufakwa ichiza. Ukuba emva Ulawulo iziyobisi wayengekho ngaphezu iiyure ezintathu ukuya kwezine, i lavage esiswini olusebenzayo, uze namalahle yokufakwa. Ukuba sele kudlule ixesha elingakumbi, unyango yenziwa unaphakade, apho kusetyenziswa dialysis (nyulu igazi kidney), diuresis (ukufumana womchamo), unyango nomqondiso.
Uluvo izigulane kwi ichiza
Uluvo izigulane ezithatha ichiza "fluconazole" kunokuba antsonkothileyo. Iqela eyahlukileyo zezigulane bonelisekile kakhulu kunye neziphumo zonyango. Ukuba esi sifo awusebenzisi, ngoko nomphumela ngokukhawuleza kwaye idla kwanele nedosi enye ye-150 mg. Kunye nemali overstrains eli chiza ayikho kakhulu xa ucinga ukuba engange ngaphakathi 250 capsule ezixabisa iziyobisi "Flucostat". Price (analogue ziqulathe ukwimo enye esebenzayo) of the philisi "fluconazole" umangale - ukusuka engange-15 ukuya kwi-30 (150 mg).
Nakuba kunjalo, kukho iqela abathengi basabela kakubi iziyobisi bulula. Ngokuqhelekileyo, zohlalutyo olunjalo zinxulunyaniswa iziphumo ebezingalindelekanga eyahlukahlukeneyo ubungnqongqo. Umntu wabonakala irhashalala, ephelekwa ukurhawuzelela kakhulu, nto leyo ixesha elide abazange baphumelele. Ezinye izigulane sele ekunyango lwe thrush, wakhalaza malunga yokuphazamiseka iphecana zesisu. Ipesenti encinane kwezigulane kweziyobisi nje swi nga pfuna. Mhlawumbi, abantu ukumelana (sifo, ukumelana) ukuya into esebenzayo.
uluvo isiqinisekiso
market zoxubo Modern ibanzi kwaye akhe ukuqonda Ukwandiswa kunye ubuqili ungakwazi kuphela ugqirha enobuchule namava. Kwaye oku iphathelene naliphi na iyeza, ukuba ngaba zentliziyo okanye yeenkqubo zengqondo, zengqondo kunye kwi-, internal medicine okanye bamazinyo. Mpilweni yokuphila nesondlo, eziphilayo embi kunye nonyango lwazo zonke izifo ukuba abacinezeli umzimba womntu, iziyobisi ezintsonkothileyo mihla kungabangela imbonakalo zizifo ezinzwaneni. Apha, igama lokugqibela kufuneka uhlale ugqirha, ukuqesha ukulungiselela unyango fungal usulelo iziyobisi "fluconazole" (nelo ukuba "Flucostat" atshiphu, kodwa akukho olusebenzayo ngaphantsi) okanye ukunikela ingqalelo kwezinye arhente amayeza nokubola.
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