Zempilo, Amalungiselelo
Analog "Trental" ku ampoules. "Trental": ezibonisa ukusetyenziswa, imfundiso
Kubo bonke ubomi mihla babonisele iingozi ezahlukeneyo. Phakathi kwazo, asiyiyo inxalenye zincinane sifo ukuthatha imiyalelo ezahlukeneyo, ubunzulu kunye nokuphelela. A ukufa ezinxulumene izifo nemithambo yegazi ngokubanzi usesikhundleni ephambili ehlabathini.
Nakuba kunjalo, inzululwazi yanamhlanje na ukuma. Izazinzulu, biochemists baye nokuqhubeka ukusebenza ekuvelisweni amachiza amatsha ukuba umntu kunceda ukuze aphumelele ekulweni isifo sentliziyo kunye imithambo yegazi. Elinye iqela imithi ezinjalo, ezibalulekileyo unyango entsonkothileyo kakhulu angioprotectors. Iziyobisi kweli qela luphawulwa umsebenzi phezulu nxamnye inkantsi ukususwa nokukhuthaza vasodilation, ukuphuculwa microcirculation, ekhokelela iimpawu eziqhelekileyo rheological igazi permeability nemithambo. Ukusebenzisa amayeza-angioprotectors kunciphisa nokudumba inyama ukutya kunye neenkqubo ukuvuselela. Ukusetyenziswa kwezi kweziyobisi eli qela ezifumaneka unyango yeendidi ezahlukeneyo angiopathy - seswekile, samathambo kunye samathambo, yegazi, iingxaki imithambo (varicose, ukuxinana kunye nokudumba), izilonda lwemithambo, nezinye izinto ezimbi efanayo.
Amaninzi, ukuze kuliwe iingxaki abasebenzi bezempilo ukumisela "Trental" (analogue beziyobisi, ngasendleleni, kukho kakhulu afikelelekayo ngaphezulu).
kuqamba leqela lendlela nemilo lokuvelisa
Eyona nto ephambili esebenzayo "Trental" i pentoxifylline. Abathengi medicament iyafumaneka iintlobo ezintathu Ukwakha: iipilisi (nganye 100 okanye 400 mg of pentoxifylline) kwaye njengesisombululo ukuba isitofu xa ampoules of ml-5 (1 ml - 20 mg of esisebenza). Ngako oko, a analog endaweni "Trental" ziphuhliswe lusekelwe pentoxifylline kunye iidosi efanayo (100 no 400 mg).
Pharmacodynamics angioprotectors
Pentoxifylline (component omkhulu "Trental") uphucula iimpawu rheological egazini, nto leyo viscous ngaphantsi nepeni. Kwakhona, le nto kuthintela zegazi kuyondelelaniswe ngokugqithiseleyo, ukhuthaza vasodilation. Ngenxa yoko, umgangatho ukuphucula microcirculation fluid zebhayoloji zomzimba (kuquka ubuchopho), kunokwenzeka kunye amathuba aphezulu ukuthintela thrombosis kunye neempahla sklerotirovanie.
Umzekelo, "Trental 400" (analogs yalo ngomlinganiselo ofanayo) kuphucula ejikelezayo kwiindawo apho ejikelezayo kuphazamisekile. Ingaba emzimbeni womntu isiphumo vasodilator myotropic (nangona buthathaka, kodwa kukho), inegalelo yokwanda kancinane iimpahla coronary. therapy kudityaniswe ukusetyenziswa kweli chiza iphucula ngokubonakalayo umfanekiso iziganeko cerebrovascular. Ukuba isigulane unesifo nakweyiphi umthambo peripheral izilonda occlusive (umz, ekuqhwaleleni), impumelelo unyango lungabonakaliswa ukwandisa umgama xa ehamba, yokuduka uxhuzula kwi namathole ngexesha sasebusuku kunye nokungabikho iintlungu yedwa.
Ubungqina obubonakalayo buxela
Le medicament "Trental" ebonisa ukuba isicelo (analogs kufuneka iimpembelelo ezifanayo emzimbeni) lo ezahlukahlukeneyo noko. Okokuqala, oko ukuphazamiseka kwegazi. Ichiza athathiweyo ukuphelisa imiphumo ngenxa yamafutha yobuchopho (nesiyezi, ukulahlekelwa inkumbulo, ukungakwazi ukunikela ingqalelo), isifo sentliziyo kobuchopho, kunye neemeko post-stroke.
Faka "Trental" analogs iziyobisi eboniswe ukuphazamiseka yegazi-flow imithambo yoluvo nendalo atherosclerotic lunomahluko trophic (izilonda trophic, babe). Nangempumelelo ke kufanelekile ukuyisebenzisa ukuphazamiseka ejikeleza medicament ocular, yegazi, utshintsho kunye iimpawu yamehlo ezenzeka ngexesha ezimbi nemithambo indlebe yangaphakathi imbono ukuhla eziviwayo kunye.
Eboniswe eli chiza kwaye ezimbi yomqolo, ezibandakanya ezifana ukutshatyalaliswa njenge stroke spinal, yegazi, ngomqolo semithambo, radiculitis, osteochondrosis, yamophula kunye nokwenzakala spinal zomlomo wakhe, ankylosing spondylitis.
Ukusebenzisa angioprotectors contraindicated?
Nawuphi angioprotector - analogu "Trental" (kwakunye, kwaye ngokwalo "Trental") - ayikwazi ukwamkela izigulane hypersensitivity kakhulu pentoxifylline, ezinye methylxanthines (pentoxifylline - ithe xanthine) okanye nayiphi na lokufaka akhoyo kule fom ukukhululwa ezifunyenweyo (tablets, iinaliti ). ukusetyenziswa azamkeleki eli qela iziyobisi ukopha enkulu na imvelaphi (pentoxifylline liyancipha viscosity igazi), hemorrhages kwi retina iliso, ingqondo, kwimo iqhosha etsolo engabalulekanga kunye nexesha ukusilela intliziyo. Ngaba contraindicated ukuba ogulayo hypotension (eliphantsi igazi uxinzelelo), sezintso ukungaphumeleli kunye wesibindi, izilonda sisilonda esiswini kunye duodenum 12. Kwimeko zongenelelo zoqhaqho "Trental" kunye analogs yayo musa ukumisela phambi kwiveki emva kotyando.
abantwana Contraindicated "Trental" (nelo kakhulu) kunye abafikisayo abangaphantsi kweminyaka eli-18 ubudala, abasetyhini abakhulelweyo kunye noomama zokonga.
ziphumo bezingalindelekanga kunokwenzeka ukuba ekufumaneni angioprotectors
Kuba naziphi angioprotectors ( "Trental" analogue) yemiyalezo sichaza iziphumo ebezingalindelekanga kunokwenzeka ukuba ngokufuthi, kodwa oko akwenzeki. Ngomhla inxalenye iphecana zesisu esiswini kungabangela intlungu, isicaphucaphu, labona ukugabha, ukuqhina, isisu esihambisayo, okanye alternation ezi States.
Nemithambo yegazi nga ndizikhumbuze ukuhlaselwa angina (esifubeni compressive iintlungu unxibe nature elifutshane-term), tachycardia, hypotension (uxinzelelo lwegazi lisibekele). ziyabagulisa ezifana ukurhawuzelela, ebuhlungu kunye nesiyezi, nokudumba angioneurotic, ukothuka anaphylactic. Ukongezelela, "Trental" analogue (ncomo yabathengi yazisa ngayo) ngamanye amaxesha baxabane ezifana ukuphazamiseka ebuthongweni-kuvukwe, ukwanda uvalo, ukuxhuzula, ukungaboni.
Ukuba kuvela ezi mpawu zingasentla, ukusetyenziswa "Trental" kufuneka ayeke, funa uqwalaselo lwamayeza, ngamanzi isisu. Ukuba kuyimfuneko, sebenzisa amayeza nomqondiso.
Ukuba amanyathelo afanelekileyo ukubuyisela imeko engasetyenziswa, amathuba ukwenzeka kwezi mpawu zilandelayo:
- nezisu kunye nokugabha "amabala ikofu" (umqondiso wokuba asakhasayo ukopha esiswini);
- kwehliswe kwezalathisi uxinzelelo wegazi;
- nokuqiniswa nesiyezi;
- ivela syncope;
- yombono;
- ukwanda iqondo lobushushu emzimbeni.
Ngophuhliso ezi mpawu kuyimfuneko ukuba iphume esiswini, iziyobisi unyango kwangumqondiso kwaye sukulibala ngemfuneko isicelo kwiimeko ezinjalo nezifunxi.
ngeedosi kakhulu: iziqhamo, amanyathelo ukuhlangabezana nazo
"Trental" ngamachiza ndlongondlongo ngokwaneleyo kwaye libanda, kunokuba naxa ingumbandela ozaliswe ziziphumo emibi. Iimpawu ezibonisa lokufumana amathamo amakhulu medicament, ukuba nesiyezi, isicaphucaphu, hypotension (ngokuwa uxinzelelo lwegazi), tachycardia (izinga intliziyo ukwanda), arrhythmia (ukubetha kwentliziyo kakubi), isikhumba ukuba bomvu, ukungabikho zingqondweni, unditsho, kuthibaza. Ukuba ucingela kukho libanda, "Trentalom" kufuneka uyeke ukuthatha kwaye ufune uncedo lonyango lobungcali. Unyango kule meko ijonge sokulondoloza kwinqanaba uxinzelelo lwegazi kunye nokusebenza zokuphefumla. Ukuba ukuxhuzula abakhoyo, ngenxa ukususwa zabo zisetyenziswa diazepam.
Xa iimpawu zokuqala ulapha kwemfuneko (isicaphucaphu, ukubila, cyanosis) eziyimfuneko ukubonelela indawo esezantsi intloko nomzimba ongasentla. ingqalelo ekhethekileyo kufuneka ihlawulwe ngokuma.
Analogs "Trental" emacwecweni
Ukuba ukhetha i analogu ilungileyo "Trental" emacwecweni, ngokoluvo iingcali ezininzi izigulane ziya idibane kumayeza "Agapurin". Indawo wokukhutshwa kwayo iSlovakia, kodwa nangona ngemvelaphi ngaphandle, kuba ixabiso iyafumaneka kuluntu jikelele kunye ezahlukeneyo kumanqanaba yengeniso. Ezikhoyo "Agapurin" kwi iidosi ezintathu - 100, 400 no-600 mg into esebenzayo.
Saziwa kakuhle ukulungiselela "kunamandla", nto leyo analog "Trental". Okubangel 'umdla kukuba, eli chiza nayo iyafumaneka ne nedosi ye-600 mg isithako esebenzayo. Amayeza kunye ne nedosi ye-pentoxifylline nga ngempumelelo nangokufanelekileyo ukujongana kwezifo ezinzima kakhulu ezinxulumene ejikeleza kakuhle. abasebenzi bezempilo "kunamandla" badla ezimiselweyo angiopathy seswekile, yegazi, imithambo yegazi Palsy zokusebenzisa ilahleko ukuva nomsindo isifo semithambo. Isiphumo HIV zisebenzisa i "kunamandla" enokwen- ukuhlaselwa ezidlulayo kobuchopho, xa sokubuyisa ixesha ekuphulukenwe nalo emva iposi engabalulekanga, ekulweni iingxaki cerebrovascular kunye nesifo Raynaud kaThixo. Effective le analogu "Trental 'emacwecweni kwaye kwiimo ukusilela acute kunye esingapheliyo yobonelelo yegazi retina iliso kunye.
Kukho analogue of "Trental", kwaye kwezinye lidle eyona nto ephambili esebenzayo. 200 no 400 mg pentoxifylline ziqulathe imithi ezifana "Trenpental", "Pentamon", "Pentilin" yaye "Pentilin Forte", "Pentomer", "Pentogeksal", "Pot", "Fleksital". Olu luhlu kusenokwenzeka ukuba uqhubeke.
Nangona kunjalo, le analogu yayixabisa "Trental" - kukuthi, ngaphandle kwamathandabuzo, "Pentoxifylline." ukukhulula ifomu xa kufikwa iipilisi - 200 no 400 mg pentoxifylline. Le medicament kufuneka bazi ukuba, ukongeza ethethelela ifuthe "Trentalu", eli chiza ingenza i-meningitis aseptic, paresthesia, iingcangcazela, nemibono, hepatitis cholestatic. Kwakhona kwezinye izigulane emva kokufumana "Pentoxifylline 'ukuze abonakale owomileyo umqala, unxano, lacrimation, lungakho okanye utshintsho ekwaneliseni iminqweno incasa. Abasebenzisi zinqabile, kodwa akhalaze ukubonakala conjunctivitis, laryngitis, earache. Ngaphezu koko, le elingana Russian "Trental" ezenza ofanelekileyo anaemia, ukopha ngegalelo lazo iimpahla cutaneous, ityhefu epidermal necrolysis.
Analogs "Trental" Inaliti
Kwiingozi ezimasikizi, xa kukho imfuneko lwezitofu, ngokuqhelekileyo abasebenzi bezempilo bakhetha imixube ezifana "Pentilin", "Lattre" (uhlobo lwe iimela), "Agapurin", "Pentoxifylline." Le bioavailability zonke ezi machiza idla kwi 98%. "Agapurin" - nelo ukuba "Trental" kwi ampoules - luqhele ukusetyenziswa kwiimeko ezininzi kakhulu ejikeleza yobuchopho, kunye imvelaphi angiopathy seswekile. Enye indawo yesicelo "agapurin"-ziphene - kwisimo izigulane emva yesifo sentliziyo, ukufa kwamalungu omzimba, kobuchopho.
Ngokufuthi lisetyenziswa "Pentilin", njengoko i-analogue of "Trental". Iingcali zikholelwa ukuba oku kulungiselelwa ixabiso elihle lemali.
imfuno umthengi lowo isisombululo ukuba ukumnika "Lattre". Ichiza ifumaneka iidosi ezintathu - 100, 200 no-400 mg. iziganeko Eminye ezingalunganga yinqobo "Trentalu" okwaziyo ukumqumbisa uphuhliso leukopenia, thrombocytopenia, pancytopenia.
Ngokubanzi, ukuba ufuna ukukhetha analogu "Trental 'ukuba isitofu okanye iimela, isiqhelo babe ngolu hlobo lulandelayo: kuqala," Pentoxifylline "njengoko umnini ixabiso eyona ndlela, ngoko" Pentilin ", apha" Latro "njenge medicament, kunye kuluhlu olubanzi yeziphumo emzimbeni womntu . Zonke ezi analogs kuba kukulungele kanye ixabiso ngaphezu "Trental", yaye bioavailability kuzo iyafana naleyo "Trental", yaye ngamanye amaxesha ngaphezulu.
Nomthamo iirejimeni of "Trental" kunye analogue yayo
azipilisi "Trental" ithathwa ngomlomo, ngaphandle ukuhlafuna okanye ezidilikayo. Yenze emva kwesidlo, amaxesha 2-3 ngosuku. Izikali - kuxhomekeke imiyalelo igqirha ukuya - inokuba ukusuka 100 ukuya 400 mg. 1200 mg - idosi iphezulu yemihla ngemihla medicament. Driving therapy kuliyeza ukuba isigulane ngasinye nomntu ngamnye iyilwe, unyango nga kuhlala naphi na ukusuka kwiiveki-2 ukuya iinyanga eziliqela.
Iinaliti "Trental" ukulungiselela (analogs kulo mzekelo angafaka isicelo isikimu eyahlukileyo) kufuneka ufakwe yegazi, bolus okanye ukumnika. Kwimeko yokuqala (jet) 1 ampoule of medicament ilawulwa ukuba imizuzu emi-5. Le nkqubo yenziwa amaxesha 1-2 emini.
Ukulungiselela ukuthontsiza, ichiza kwi imali ampoules ukusuka kwisi-1 ukuya ku-6, ugalelwe saline okanye 5 ekhulwini iswekile. Ithuba Ukuqaliswa kwalo mxube - up to iyure-1. Beka dropper namaxesha 1-2 emini. Ubuninzi kwiintsuku amathontsi faka kuvunyelwe 1200 mg medicament (ampoules 12).
Angioprotector "Lattre" - nelo ukuba 'Trental "kunye kuluhlu olubanzi amanyathelo - isetyenziswe ukunyanga kwi inkqubo yayo. Amaninzi kusetyenziswa lolawulo efakwa. Ikhosi ye unyango isigulane ngamnye liphuhlisa ugqirha ofanelekayo, kuthathelwa ingqalelo ubunzima bomzimba kunye ubuzaza imeko yakhe mntu. Imvaba "Latro" (200 ml) ukuba isitofu ibe ukuthontsiza iphuma iiyure 1.5-3. Ukuba akukho iziganeko ezibi lungenzeki, kunokwenzeka ukuba ukwandisa umthamo ukuya 400-500 ml medicament.
Ukongeza, amachiza analogu "Trental" ukusetyenziswa ngokuvunywe abantwana abangaphantsi kweminyaka eli-12 ubudala. Kulo mzekelo, ithamo kancinane olusebenzayo ibalwa kwekilogram ubunzima bomzimba yomntwana ngamnye. Amaninzi, abantwana ifuna ukufumana 5 mg iziyobisi kwekilogram ubunzima bomzimba ngalinye.
Imibono malunga "Trentale" kunye analogue zayo kwizigulane kunye nabasebenzi bezempilo
Njengalo naluphi na Togu "Trental" kwaye ngokwalo medicament olusebenzayo kwezifo ngokwaneleyo ezimbi kwi kwegazi. Nakuba kunjalo, iziphumo ebezingalindelekanga kweziyobisi ezinjalo lukhulu. Inani elaneleyo izigulane ezithatha angioprotectors (kwaye "Trental" ingakumbi) ngethuba elisusela kokuvuselelwa emva kokuhlaselwa sentliziyo nestroke. Kwiimeko ezininzi, iyeza iye yaqinisekisa iimpawu kwizinga eliphezulu ichiza. Nangona maxa wambi wadibana ukubuyekeza ingxolo ezindlebeni, bawe uxinzelelo lwegazi.
Iqela olwahlukileyo izigulane, "Trental 'elawulwa ngenxa yonyango wokuva ilahleko. Uninzi reviews zezi abasebenzisi ingculaza.
Le Izimo amayeza - zomitho zisanyisa. Nakuba kunjalo, kaninzi gynecologists amisele ichiza kubafazi abakhulelweyo ukuphucula kwegazi okanye izityalo isondlo. Iqela olwahlukileyo izigulane wayalelwa ukuba "Trental" njengenyathelo lothintelo.
Ngokubanzi, ukuba "Trental" (njengoko, eneneni, naliphi na ibakala elilingana neli) ziya ingonyulwa ukhathalelo lwempilo oyingcali kunye irejimeni olufanayo unyango ziya kuphuhliswa, ngoko ke umngcipheko yeziphumo ebezingalindelekanga ziyakuncitshiswa, kwaye ichiza bonakalisa kakhulu ngempumelelo.
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