Zempilo, Amalungiselelo
"Voltaren" - udaka, lulekani iqolo, ubuhlungu bemisipha. Imiyalelo yokusebenzisa
"Voltaren" (patch) - ekunyangeni arhente kunye nokubhalwe diclofenac, zikwenze amalungu abe buhlungu, emva izihlunu. Lo patch yokuqala, aba izixhobo zonyango kunye neziyobisi.
imiphumela kwemithi
Le medicament i isiseko laphu ukuba leyo Usebenzise umaleko kwakuse equlethe diclofenac - NSAIDs abe eminyaka ezisetyenziswa kwezonyango ekunciphiseni iintlungu, ukudumba kunye ukuqina e arthropathies ukudumba, osteoarthritis, isifo samathambo kunye konzakale kwizihlunu ezithambileyo, iqolo. Icandelo Active abangaphangeliyo prostaglandin yokuqaphela, ngaloo ndlela ekufezekiseni iziphumo anti-ezithintela ukosuleleka kunye iintlungu va. Ummandla isicelo iyapheliswa iintlungu, ukuncipha kudumba ezinxulumene inkqubo komtshiso oko. Kwakhona, "Voltaren" (patch) kuphula embundwini intlungu (ngokunxulumene le ukusebenza kwayo kubhetele ukusebenzisa patch "Indomethacin", uqinisekiswe review).
Pharmacokinetics
kufumaneka ngokorhwebo maleko enamathelayo of diclofenac kwisithuba iiyure ezingamashumi amabini anesine stably ingena kulusu ukuya kumthombo intlungu. Uyondelelwano lwee- esisebenza inwebu yesihlunu usebenzisa patch "Voltaren" iyafana xa kufakwa gel "Voltaren Emulgel." Ngoko ke, singatsho ukuba ezi amachiza bioequivalent. Nge protein yintloya sibophelela 99,7% of diclofenac, kuquka albumin - 99,4%. Isiqingatha-ebomini into esebenzayo - Iiyure enye okanye ezimbini. Half-ubomi metabolites - iiyure enye ukuya kwezintathu. Kukhuthaza wenziwa ngakumbi yokuchama.
Xa izigulane umsebenzi kakuhle kwezintso, akukho ukuqokelela diclofenac kunye metabolites. Abantu abane kwesibindi nedekompensirovannym okanye kohlobo ukutya kunye kinetics ze isithako esebenzayo lwenzeka ngendlela efanayo ebantwini, ngaphandle isifo zesibindi.
Ubungqina obubonakalayo buxela
Iya ngempumelelo kunyanga "Voltaren" kwizifo ezininzi izixhobo motor. Udaka sisetyenziselwa iqolo kwimeko ezimbi sisiba mandundu kwaye ukudumba spinal (e osteoarthritis, sciatica, sciatica, lumbago), iintlungu kwezihlunu, evela nokulatyuza yokwenzakala, komsipha, nemivumbo, kunye neentlungu elidityanelweyo osteoarthritis, isifo samathambo. Phakathi kwezinye izinto, oku kusetyenziswa ukuphelisa ukufukuka kunye ukudumba amalungu kunye izicwili ezithambileyo kuzo izifo samathambo (bursitis, tenosynovitis, izilonda izicwili periarticular).
ifomu idosi nokwakheka
Le patch ngokumila ebuxande elintlangothi ajikelezayo, iqulathe isiseko ye ipholiyesta beige-obugolide, olusetyenziswa ngokufanayo maleko enamathelayo kunye eliqhelekileyo livumba elithozamisayo (umbala ngcina umphezulu inokuba ukusuka ezingenambala ube tyheli). Umaleko ngcina wambu zokukhusela top umboniso seplastikhi esitransparenti ukusikwa ezimbini ezinqamlezayo (ngomhla enye kumgca esimfaneleko i). On the ifilimu yokuchaza ebonisa indlela kuyimfuneko ukuba asuse kumphezulu ngcina.
Kukho iintlobo ezininzi arhente zonyango ochazwe "Voltaren". Patch elakhiwa 15 okanye 30 mg diclofenac sodium. Kweli nqaku, eziquka-15 mg isithako esebenzayo ineenkalo 70 x 100 eemilimitha, kwaye i-30 mg - 100 x 140 mm. izithako Minor benza methylpyrrolidone, efirizirovannaya gum, citric acid, levomenthol, polyisobutylene, propylene ethers esters okunamafutha acid, izoprenstirol copolymer butylhydroxytoluene, ngokusekelwe imicu ipholiyesta, mercaptobenzimidazole, iparafini elulwelo, a protective umboniso eyenziwe ipholiyesta.
Indlela yokwenza isicelo nesiziba "Voltaren '? Imiyalelo. inani
Le patch lusetyenziswa ulusu ngohlobo izicelo. Kufuneka njo kwindawo buhlungu, yaye musa adubule iiyure ezingamashumi amabini anesine. Per ebusuku yaye bavunyelwe ukuba basebenzise imveliso enye kuphela. Ngokutsho manani, xa izigulane zithandwa kakhulu ukuphiliswa patch "Voltaren". Ingxelo evela kwabo ukuyisebenzisa uzijonga njengento eluncedo kwi kwindawo yokuqala ukuya lula isicelo off. Izigulana nazo ziyakhuthazwa ukuba sifakiweyo awubonakali phantsi kwengubo (ngenxa yokuba abavelisi kwenze ultra-ezingcakacileyo, ibala). Ukuba sisilonda esidumbileyoesingaphakathi olubanzi, kufuneka usebenzise ubungakanani imveliso i-140 x 100 iimilimitha. Kuba unyango yokwenzakala zeethishu soft isicelo nesiziba kufuneka iintsuku kungekho ngaphezulu kwe elinesine, izifo amalungu kunye nezihlunu - hayi ngaphezu kweentsuku ezingamashumi amabini ananye (ngaphandle kokuba ugqirha icwangcisa a mode). Ukuba imeko uhlala enye, okanye mandundu emva kweentsuku ezisixhenxe unyango, kufuneka uyeke ukusebenzisa ichiza aze adibane lweengcali icebiso ngendlela yokwenza oku.
Le patch ngesi Pharmacy embodiments eziliqela. Ngenxa yoko, imveliso iqulethe 15 neemiligram diclofenac ziya kuthengiswa upakisho zizele-2 okanye 5. Kwimeko yokuqala, ixabiso isusela kwi-avareji engange-125 ukuya 145, owesibini - ukusuka engange-270 ukuya 315. Patch equlathe milligrams 30 diclofenac, kuthengiswa iipakethe amaqhosha 2. Indleko ezikhemisti ezahlukeneyo iyahluka ukusuka engange 205 ukuya 220. Yonke imveliso abhijelwe iingxowa ngefoyile ye-aluminiyam, mvisiswano leyo, kwelinye icala, zingafakwa kwiibhokisi kwikhadibhodi. Ukunikezela lokumiselwa ukuthenga ichiza efunekayo.
imiphumela emibi
Imiphumo ezimbi ukuze aphuhlise phezu yangasemva isiziba "Voltaren", ngokusisiseko koko obubonakala ulusu entsimini lwesicelo (njenge umthetho, ukuba ichazwa ephakathi, kunye idlule). Ngoko ke, kwezinye izigulane, kukho papules, ukudumba, ukurhawuzelela, vesicles, erythema, bechuba, irhashalala, nerhashalala. Kwiimeko ezinqabe kakhulu, kukho bullous dermatitis. Kwabanye abantu (ngamaxesha ambalwa) ezivela ekusetyenzisweni kwe patch kwenzeka pustular irhashalala, photosensitivity reaction, ngokubanzi amaqhakuvana eluswini, negazi ezifana ukuhlaselwa sisifo sombefu, bronchospasm, urticaria, angioedema.
Izimo
Phambi hypersensitivity ukuya diclofenac okanye namanye amacandelo ezikhoyo ekwakhiweni kufuneka sisebenzise medicament. Kukwacetyiswa kwakhona ukuba isicelo eso sifakiweyo, abo sinotyekelo nokuthimliswa kakhulu, ukuhlaselwa isifuba inyumoniya, irhashalala, wenza unyango kunye acetylsalicylic acid okanye ezinye NSAIDs. Ukusetyenziswa imveliso contraindicated abantwana abangaphantsi kweminyaka elishumi elinesihlanu ubudala. Akukho mfuneko uncamathelise nesiziba kwi ngamayelenqe apho isikhumba punctured ezikuyo. Ngenyameko kusetyenziswa phambi ilunga-ezilinyaziweyo izitshanguba ye phecana zesisu, ukusilela intliziyo, iintlobo ezinganyangekiyo ukuphazamiseka kakhulu ezintso okanye isibindi, porphyria hepatic (in exacerbation).
Sebenzisa ngethuba lokukhulelwa zisanyisa
Ngenxa yokungabikho data kwi ukuba i "Voltaren" patch neziphumo ezibi ekukhuleni kosana olungekazalwa ngethuba lokukhulelwa, kwaye nokuba ludlulele ubisi lwebele, abasetyhini abakhulelweyo kunye zokonga kufuneka bakuphephe ukusetyenziswa kwayo.
Libanda, kunye nentsebenziswano kunye namanye amayeza
Ngenxa yokuba ukusetyenziswa yangaphandle kuqulunqo medicament nokufunxwa izithako ezisebenzayo iphantsi kakhulu, i libanda wayo basuswe.
Nesicelo ngaxeshanye ityatyekwe neziyobisi ezibangela photosensitivity, umphumo wokugqibela kwengeniso. Intsebenziswano kunye namanye amachiza nokuba ukubaluleka lwezonyango, akwenziwanga ichazwa.
oyi
Umele ungafaki amacandelo yokusebenza umnikelo le ngcina ngomaleko patch, inwebu yangaphakathi okanye amehlo. Le mveliso uvumelekile ukuba ukunamathelisa pokrvy kuphela ezingonakalanga, ukusetyenziswa kwayo kwimihlaba kunye amanxeba avulekileyo akwamkelekanga. Xa usebenzisa isiziba "Voltaren" ixesha elide kakhulu, kukho umngcipheko wokuba ngayo ezibi lwenkqubo. Ukuba ukongeza imveliso echazwe isicelo eminye imithi eziqulathe diclofenac kuyimfuneko ukuqwalasela umxholo wenkqu inxaxheba patch, yaye singadluli bobude ukuba idosi yemihla ngemihla (kuba milligrams 150). Izifundo oluqhubekayo aye abonisa ukuba izinga reactions lengqondo xa usebenzisa oomatshini kunye nokuqhuba le fomu umthamo ichiza "Voltaren" lungenasiphumo. Ubude bethuba ubomi patch xa zigcinwa kwi bezifakwe kuyo, kwakunye lobushushu elingadluliyo 25 Degrees Celsius iminyaka emibini.
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